SCHEMBL4904568

SCHEMBL4904568

COc1cc(N2CCn3cc(-c4ccc(Cl)cc4)cc3C2=O)ccc1OCCNC(=O)O

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 16/20 0.46
KCNH2 Q12809 1/20 0.46
HTR2A P28223 3/20 0.42
HTR2C P28335 3/20 0.42
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14458780 0.90 MCHR1 (0.48) MCHR1KCNH2HTR2AHTR2CHTR2B
SCHEMBL1930352 0.90 MCHR1 (0.43) MCHR1KCNH2HTR2AHTR2CHTR2B
SCHEMBL12532018 0.86 MCHR1 (0.47) MCHR1KCNH2HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL1928535 0.85 MCHR1 (0.47) MCHR1KCNH2HTR2AHTR2CHTR2B
SCHEMBL1928022 0.84 MCHR1 (0.49) MCHR1KCNH2HTR2AHTR2C
SCHEMBL1930223 0.84 MCHR1 (0.51) MCHR1KCNH2HTR2AHTR2CHTR2B
Trifluoroacetic Acid SCHEMBL1929462 0.84 MCHR1 (0.57) MCHR1KCNH2HTR2AHTR2CHTR2B
SCHEMBL12531954 0.83 MCHR1 (0.62) MCHR1KCNH2HTR2AHTR2CHTR2B
Trifluoroacetic Acid SCHEMBL1931079 0.83 MCHR1 (0.52) MCHR1KCNH2HTR2AHTR2CHTR2B
Trifluoroacetic Acid SCHEMBL1930599 0.83 MCHR1 (0.45) MCHR1KCNH2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987039-A2 MELANIN CONCENTRATING HORMONE RECEPTOR-1 ANTAGONISTS Brystol-Myers Squibb Company (US) 2008-11-05 EP disclosed
WO-2007092416-A2 MELANIN CONCENTRATING HORMONE RECEPTOR-1 ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-08-16 WO disclosed