SCHEMBL4915641

SCHEMBL4915641

O=C(C1CCN(Cc2ccn(-c3ccc(C(F)(F)F)cc3)c2)CC1)N1CC=C(c2ccc(Cl)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 20/20 0.56
KCNH2 Q12809 15/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4923627 0.89 MCHR1 (0.64) MCHR1KCNH2
SCHEMBL5316462 0.77 MCHR1 (0.65) MCHR1KCNH2
Chlorolithium SCHEMBL4922637 0.76 MCHR1 (0.62) MCHR1KCNH2
SCHEMBL5322252 0.75 DRD4 (0.60) MCHR1KCNH2
Hydrochloric Acid SCHEMBL27710070 0.75 MCHR1 (0.63) MCHR1KCNH2
SCHEMBL4924154 0.72 MCHR1 (0.86) MCHR1KCNH2
SCHEMBL4925599 0.72 MCHR1 (0.59) MCHR1KCNH2
SCHEMBL4925438 0.72 MCHR1 (1.00) MCHR1KCNH2
SCHEMBL5316946 0.71 MCHR1 (0.72) MCHR1KCNH2
SCHEMBL4925981 0.71 MCHR1 (0.56) MCHR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080306055-A1 Heterocyclic Mchr1 Antagonists And Their Use In Therapy ASTRAZENECA AB (SE) 2008-12-11 US claimed
EP-1831194-A1 HETEROCYCLIC MCHr1 ANTAGONISTS AND THEIR USE IN THERAPY AstraZeneca AB (SE) 2007-09-12 EP claimed
WO-2006068594-A1 HETEROCYCLIC MCHr1 ANTAGONISTS AND THEIR USE IN THERAPY ASTRAZENECA AB (SE) 2006-06-29 WO claimed
US-20080306055-A1 Heterocyclic Mchr1 Antagonists And Their Use In Therapy ASTRAZENECA AB (SE) 2008-12-11 US disclosed
EP-1831194-A1 HETEROCYCLIC MCHr1 ANTAGONISTS AND THEIR USE IN THERAPY AstraZeneca AB (SE) 2007-09-12 EP disclosed
WO-2006068594-A1 HETEROCYCLIC MCHr1 ANTAGONISTS AND THEIR USE IN THERAPY ASTRAZENECA AB (SE) 2006-06-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080306055-A1 Heterocyclic Mchr1 Antagonists And Their Use In Therapy MCHR1, MCHR2, MC1R MCHR1 1/4885KCNH2 1440/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.