SCHEMBL4924470

SCHEMBL4924470

O=S(=O)(c1ccc(CNCc2ccccn2)cc1)N(Cc1nc2ccccc2[nH]1)C1CCCc2ccccc21

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 18/20 0.66
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
CYP2D6 P10635 2/20 0.43
CYP3A4 P08684 1/20 0.43
TAS2R14 Q9NYV8 1/20 0.43
CHRM2 P08172 1/20 0.43
DRD2 P14416 1/20 0.43
OPRM1 P35372 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4913565 0.92 CXCR4 (0.76) CXCR4CYP2D6CYP3A4CHRM2DRD2
SCHEMBL4923734 0.91 CXCR4 (0.53) CXCR4CYP2D6TAS2R14CHRM2DRD2
SCHEMBL4924464 0.85 CXCR4 (0.50) CXCR4CYP2D6TAS2R14CHRM2DRD2
SCHEMBL29823518 0.80 CXCR4 (1.00) CXCR4CYP2D6CYP3A4CHRM2DRD2
SCHEMBL1878773 0.80 CXCR4 (1.00) CXCR4CYP2D6CYP3A4CHRM2DRD2
Bromide SCHEMBL4544117 0.79 CXCR4 (0.98) CXCR4CYP2D6CYP3A4CHRM2DRD2
SCHEMBL14025556 0.78 PDE4A (0.52) CXCR4PDE4APDE4BPDE4CPDE4D
SCHEMBL4786868 0.77 CXCR4 (0.54) CXCR4PDE4APDE4BPDE4CPDE4D
SCHEMBL14025404 0.77 CXCR4 (0.58) CXCR4PDE4APDE4BPDE4CPDE4D
SCHEMBL4913569 0.76 CXCR4 (0.59) CXCR4CYP2D6CHRM2DRD2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea METASTATIX, INC. 2008-10-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea MKI67, CCNI, CDKN1A CXCR4 242/4885PDE4A 2435/4885PDE4B 2396/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.