SCHEMBL4928908

SCHEMBL4928908

Cc1nc(C(=O)N(C)CCOC(=O)C(F)(F)F)cc2c(Nc3cccc4c3CCO4)c(C(N)=O)cnc12

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.47
MTNR1B P49286 1/20 0.33
CSF1R P07333 8/20 0.33
EED O75530 2/20 0.33
SUZ12 Q15022 2/20 0.33
EZH2 Q15910 2/20 0.33
BRD4 O60885 2/20 0.32
BRD2 P25440 2/20 0.32
BRD3 Q15059 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
RBBP4 Q09028 1/20 0.32
AEBP2 Q6ZN18 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4930021 0.90 PDE4B (0.51) PDE4BMTNR1BCSF1REEDSUZ12
Trifluoroacetic Acid SCHEMBL4928901 0.89 PDE4B (0.48) PDE4BMTNR1BCSF1REEDSUZ12
Trifluoroacetic Acid SCHEMBL4929976 0.84 PDE4B (0.51) PDE4BMTNR1BCSF1REEDSUZ12
Trifluoroacetic Acid SCHEMBL4929251 0.82 PDE4B (0.48) PDE4BMTNR1BCSF1RBRD4BRD2
SCHEMBL4924230 0.81 PDE4B (0.57) PDE4BMTNR1BCSF1RBRD4BRD2
SCHEMBL4928534 0.81 PDE4B (0.59) PDE4BMTNR1BCSF1REEDSUZ12
Trifluoroacetic Acid SCHEMBL4928658 0.80 PDE4B (0.47) PDE4BMTNR1BCSF1RBRD4BRD2
Trifluoroacetic Acid SCHEMBL4920920 0.79 PDE4B (0.45) PDE4BCSF1REEDSUZ12EZH2
SCHEMBL5765629 0.78 PDE4B (0.51) PDE4BMTNR1BCSF1R
Trifluoroacetic Acid SCHEMBL4930184 0.78 PDE4B (0.47) PDE4BMTNR1BCSF1REEDSUZ12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080146563-A1 1,7-Naphthyridines as Pde4 Inhibitors GLAXO GROUP LIMITED 2008-06-19 US claimed
US-20080146563-A1 1,7-Naphthyridines as Pde4 Inhibitors GLAXO GROUP LIMITED 2008-06-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080146563-A1 1,7-Naphthyridines as Pde4 Inhibitors PDE4A, PDE3B, PDE4B PDE4B 3/4885MTNR1B 694/4885CSF1R 4095/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.