SCHEMBL4942464

SCHEMBL4942464

O=c1[nH]cccc1-c1noc(-c2cc(O)c(O)c([N+](=O)[O-])c2)n1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
COMT P21964 1/20 0.49
RXFP1 Q9HBX9 1/20 0.42
S1PR1 P21453 3/20 0.42
MAPT P10636 6/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
ALDH1A1 P00352 1/20 0.39
ABCB1 P08183 1/20 0.39
KMT2A Q03164 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
HPGD P15428 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1447624 0.79 COMT (0.60) COMTRXFP1S1PR1MAPTNPC1
SCHEMBL3586619 0.79 COMT (0.49) COMTRXFP1S1PR1MAPTNPC1
SCHEMBL3585954 0.77 COMT (0.48) COMTRXFP1S1PR1MAPTNPC1
SCHEMBL3592774 0.75 COMT (0.55) COMTRXFP1S1PR1MAPTNPC1
SCHEMBL1447281 0.75 COMT (0.55) COMTRXFP1MAPTNPC1RAB9A
SCHEMBL3580951 0.75 COMT (0.60) COMTS1PR1MAPTNPC1RAB9A
SCHEMBL1447309 0.75 COMT (0.50) COMTRXFP1S1PR1MAPTNPC1
SCHEMBL1447346 0.74 COMT (0.59) COMTS1PR1MAPTNPC1RAB9A
SCHEMBL1447306 0.74 COMT (0.52) COMTRXFP1S1PR1MAPTNPC1
SCHEMBL3586856 0.74 COMT (0.53) COMTS1PR1MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed