SCHEMBL4949162

SCHEMBL4949162

CCc1cc(-n2nc(-c3nc4cc5c(cc4[nH]3)N(C(C)C)C(=O)C5(C)C)c3c2CN(C(=O)O)C3)cc(CC)c1C(N)=O

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4948596 0.90 AURKA (0.43) AURKAAURKB
SCHEMBL4946077 0.76 ITK (0.37) AURKAAURKB
SCHEMBL4949158 0.69 AURKA (0.42) AURKAAURKB
SCHEMBL4827138 0.67 AURKA (0.40) AURKAAURKB
SCHEMBL4948961 0.67 AURKA (0.53) AURKAAURKB
SCHEMBL4965819 0.66 AURKA (0.35) AURKAAURKB
SCHEMBL4827132 0.66 AURKA (0.44) AURKAAURKB
SCHEMBL4950836 0.65 AURKA (0.40) AURKAAURKB
SCHEMBL4948278 0.65 AURKA (0.42) AURKAAURKB
SCHEMBL4891748 0.65 PAK4 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885725-B1 TRICYCLIC AZOLE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS HOFFMANN LA ROCHE (CH) 2008-09-24 EP disclosed