SCHEMBL4952241

SCHEMBL4952241

O=[N+]([O-])c1cc(-c2nc(C(O)c3ccc(C(F)(F)F)nc3)no2)cc(O)c1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
COMT P21964 1/20 0.41
BRD4 O60885 1/20 0.35
TTR P02766 2/20 0.35
POLB P06746 3/20 0.34
TRPV3 Q8NET8 4/20 0.33
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
MAPT P10636 4/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3587756 0.82 COMT (0.49) COMTTTRPOLBMAPTNPC1
SCHEMBL3593513 0.80 COMT (0.47) COMTTTRPOLBMAPTNPC1
SCHEMBL4952238 0.78 TTR (0.44) COMTTTRMAPTNPC1RAB9A
SCHEMBL3587362 0.74 TTR (0.40) COMTTTRPOLBCRHBPCRHR2
SCHEMBL3588271 0.74 TTR (0.38) COMTTTRTRPV3CRHBPCRHR2
SCHEMBL3582679 0.73 COMT (0.52) COMTTTRPOLBMAPTNPC1
SCHEMBL3587929 0.71 TTR (0.38) COMTTTRCRHBPCRHR2MAPT
SCHEMBL3585954 0.71 COMT (0.48) COMTTTRPOLBMAPTNPC1
SCHEMBL3587928 0.70 TTR (0.43) COMTTTRCRHBPCRHR2MAPT
SCHEMBL3582149 0.70 COMT (0.49) COMTTTRPOLBMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed