SCHEMBL4954887

SCHEMBL4954887

COc1ccc(-c2ccc(N3CCC4CN(C)CC43)cc2)cn1

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 17/20 0.70
KCNH2 Q12809 2/20 0.58
CHRNB2 P17787 2/20 0.46
CHRNB4 P30926 2/20 0.46
CHRNA3 P32297 2/20 0.46
CHRNA4 P43681 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3058284 1.00 HRH3 (0.70) HRH3KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL3053078 0.87 HRH3 (0.71) HRH3KCNH2
SCHEMBL3058127 0.83 HRH3 (0.72) HRH3KCNH2
SCHEMBL3062819 0.83 HRH3 (0.66) HRH3KCNH2
SCHEMBL3057839 0.82 HRH3 (1.00) HRH3KCNH2
SCHEMBL3052800 0.80 HRH3 (0.70) HRH3KCNH2
SCHEMBL3053033 0.80 HRH3 (0.70) HRH3KCNH2
SCHEMBL3070874 0.79 HRH3 (0.71) HRH3KCNH2
SCHEMBL3057657 0.78 HRH3 (0.74) HRH3KCNH2
SCHEMBL3054388 0.78 HRH3 (0.66) HRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001885-A2 OCTAHYDRO-PYRROLO[3,4-B]PYRROLE DERIVATIVES Abbott Laboratories (US) 2008-12-17 EP disclosed
WO-2007100990-A2 OCTAHYDRO-PYRROLO[3,4-B] PYRROLE DERIVATIVES AND THEIR USE AS HISTAMINE-3 RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2007-09-07 WO disclosed