SCHEMBL4958437

SCHEMBL4958437

COCCCNC(=O)c1ccc(Nc2ncc(F)c(-c3cnc(C)n3C3CCOCC3)n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 13/20 0.51
CDK1 P06493 6/20 0.51
KCNH2 Q12809 5/20 0.50
JAK2 O60674 2/20 0.49
JAK1 P23458 2/20 0.49
JAK3 P52333 2/20 0.49
CDK4 P11802 4/20 0.44
CCND3 P30281 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4251212 0.99 CDK2 (0.51) CDK2CDK1KCNH2JAK2JAK1
Hydrochloric Acid SCHEMBL4249706 0.90 CDK2 (0.53) CDK2CDK1KCNH2JAK2JAK1
SCHEMBL4959333 0.88 CDK2 (0.55) CDK2CDK1KCNH2JAK2JAK1
Hydrochloric Acid SCHEMBL4250789 0.88 CDK2 (0.56) CDK2CDK1KCNH2JAK2JAK1
Hydrochloric Acid SCHEMBL4248251 0.87 CDK2 (0.54) CDK2CDK1KCNH2JAK2JAK1
Hydrochloric Acid SCHEMBL4246170 0.86 CDK2 (0.53) CDK2CDK1KCNH2JAK2JAK1
Hydrochloric Acid SCHEMBL4249609 0.86 CDK2 (0.64) CDK2CDK1KCNH2JAK2JAK1
Hydrochloric Acid SCHEMBL4245085 0.85 CDK2 (0.66) CDK2CDK1KCNH2JAK2JAK1
Hydrochloric Acid SCHEMBL4249423 0.85 CDK2 (0.58) CDK2CDK1KCNH2
SCHEMBL13879010 0.84 CDK2 (0.54) CDK2CDK1KCNH2JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945628-A1 NEW PYRIMIDINE DERIVATIVES AND THEIR USE IN THERAPY AS WELL AS THE USE OF PYRIMIDINE DERIVATIVES IN THE MANUFACTURE OF A MEDICAMENT FOR PREVENTION AND/OR TREATMENT OF ALZHEIMER'S DISEASE AstraZeneca AB (SE) 2008-07-23 EP disclosed
WO-2007040440-A1 NEW PYRIMIDINE DERIVATIVES AND THEIR USE IN THERAPY AS WELL AS THE USE OF PYRIMIDINE DERIVATIVES IN THE MANUFACTURE OF A MEDICAMENT FOR PREVENTION AND/OR TREATMENT OF ALZHEIMER’S DISEASE ASTRAZENECA AB (SE) 2007-04-12 WO disclosed