SCHEMBL495883

SCHEMBL495883

C1=CSCCN1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL31340495 0.97
SCHEMBL1829299 0.82
SCHEMBL1782650 0.67
SCHEMBL38003 0.67
Thiazolidine SCHEMBL6425125 0.63
SCHEMBL1834157 0.62
SCHEMBL3339679 0.59
SCHEMBL1829036 0.59
SCHEMBL108935 0.58
SCHEMBL15387767 0.55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 473 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4663182-A2 PROPHYLACTIC OR THERAPEUTIC AGENT FOR HYPOXIC INJURY, ISCHAEMIA-REPERFUSION INJURY AND INFLAMMATION, CELL PROTECTION AGENT FOR TRANSPLANTATION, AND BIO-PRESERVATION AGENT Scent Science International Inc. (JP) 2025-12-17 EP claimed
CN-119345196-A Preventive or therapeutic agent for hypoxia disorder, ischemia reperfusion disorder or inflammation, cytoprotective agent for transplantation, and organism preservative 脑科学香料株式会社 2025-01-24 CN claimed
CN-119112885-A Preventive or therapeutic agent for hypoxia disorder, ischemia reperfusion disorder or inflammation, cytoprotective agent for transplantation, and organism preservative 脑科学香料株式会社 2024-12-13 CN claimed
CN-119015277-A Preventive or therapeutic agent for hypoxia disorder, ischemia reperfusion disorder or inflammation, cytoprotective agent for transplantation, and organism preservative 脑科学香料株式会社 2024-11-26 CN claimed
US-20240382497-A1 PROPHYLACTIC OR THERAPEUTIC AGENT FOR HYPOXIC INJURY, ISCHAEMIA-REPERFUSION INJURY AND INFLAMMATION, CELL PROTECTION AGENT FOR TRANSPLANTATION, AND BIO-PRESERVATION AGENT SCENT SCIENCE INTERNATIONAL INC. (JP) 2024-11-21 US claimed
US-20230293542-A1 SENSORY STIMULATING PSYCHOTROPIC DRUG KANSAI MEDICAL UNIVERSITY (JP) 2023-09-21 US claimed
CN-116437916-A Sensory stimulation mental medicine 学校法人关西医科大学 2023-07-14 CN claimed
EP-4190325-A1 SENSORY STIMULATING PSYCHOTROPIC DRUG Kansai Medical University (JP) 2023-06-07 EP claimed
US-20230149417-A1 PROPHYLACTIC OR THERAPEUTIC AGENT FOR HYPOXIC INJURY, ISCHAEMIA-REPERFUSION INJURY AND INFLAMMATION, CELL PROTECTION AGENT FOR TRANSPLANTATION, AND BIO-PRESERVATION AGENT SCENT SCIENCE INTERNATIONAL INC. (JP) 2023-05-18 US claimed
US-20230149420-A1 ANTI-INFLAMMATORY IMMUNOENHANCER SCENT SCIENCE INTERNATIONAL INC. (JP) 2023-05-18 US claimed
EP-1551811-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS VANILLOID RECEPTOR LIGANDS Amgen Inc. (US) 2005-07-13 EP claimed
EP-1542692-A1 AMINO-PYRIDINE, -PYRIDINE AND PYRIDAZINE DERIVATIVES FOR USE AS VANILLOID RECEPTOR LIGANDS FOR THE TREATMENT OF PAIN Amgen Inc. (US) 2005-06-22 EP claimed
EP-1463714-A2 VANILLOID RECEPTOR LIGANDS AND THEIR USE IN TREATMENTS Amgen Inc. (US) 2004-10-06 EP claimed
US-20040152690-A1 Vanilloid receptor ligands and their use in treatments AMGEN INC. 2004-08-05 US claimed
US-20040082780-A1 Vanilloid receptor ligands and their use in treatments AMGEN, INC. 2004-04-29 US claimed
WO-2004035549-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS VANILLOID RECEPTOR LIGANDS AMGEN INC. (US) 2004-04-29 WO claimed
US-20040038969-A1 Vanilloid receptor ligands and their use in treatments AMGEN, INC. 2004-02-26 US claimed
WO-2003099284-A1 AMINO-PYRIDINE, -PYRIDINE AND PYRIDAZINE DERIVATIVES FOR USE AS VANILLOID RECEPTOR LIGANDS FOR THE TREATMENT OF PAIN AMGEN INC. (US) 2003-12-04 WO claimed
US-20030195201-A1 Vanilloid receptor ligands and their use in treatments AMGEN INC. 2003-10-16 US claimed
WO-2003049702-A2 VANILLOID RECEPTOR LIGANDS AND THEIR USE IN TREATMENTS AMGEN INC. (US) 2003-06-19 WO claimed