Troglitazone

Troglitazone

SCHEMBL4959

Cc1c(C)c2c(c(C)c1O)CCC(C)(COc1ccc(CC3SC(=O)NC3=O)cc1)O2

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPARG

The experimentally established mechanism targets of Troglitazone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG known ✓ P37231 8/20 0.50
MEN1 O00255 2/20 0.64
MAPT P10636 2/20 0.64
KMT2A Q03164 2/20 0.64
TDP1 Q9NUW8 2/20 0.64
CYP3A4 P08684 2/20 0.56
ALDH1A1 P00352 1/20 0.56
TP53 P04637 1/20 0.56
CYP1A2 P05177 1/20 0.56
HPGD P15428 1/20 0.56
ALOX15 P16050 1/20 0.56
TSHR P16473 1/20 0.56
HSD17B10 Q99714 1/20 0.56
FFAR1 O14842 5/20 0.45
PPARA Q07869 2/20 0.45
HRH3 Q9Y5N1 1/20 0.43
RXRA P19793 1/20 0.42
MPC2 O95563 2/20 0.41
CYP2C8 P10632 2/20 0.41
CYP2C9 P11712 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Troglitazone SCHEMBL12496814 1.00 MEN1 (0.64) MEN1MAPTKMT2ATDP1CYP3A4
Troglitazone SCHEMBL30050392 1.00 MEN1 (0.64) MEN1MAPTKMT2ATDP1CYP3A4
Troglitazone SCHEMBL8496660 1.00 MEN1 (0.64) MEN1MAPTKMT2ATDP1CYP3A4
Troglitazone SCHEMBL29349864 1.00 MEN1 (0.64) MEN1MAPTKMT2ATDP1CYP3A4
Troglitazone SCHEMBL1536757 1.00 MEN1 (0.64) MEN1MAPTKMT2ATDP1CYP3A4
Troglitazone SCHEMBL5672808 1.00 MEN1 (0.64) MEN1MAPTKMT2ATDP1CYP3A4
Troglitazone SCHEMBL21630 1.00 MEN1 (0.64) MEN1MAPTKMT2ATDP1CYP3A4
Troglitazone SCHEMBL15888838 1.00 MEN1 (0.64) MEN1MAPTKMT2ATDP1CYP3A4
Troglitazone SCHEMBL5672813 1.00 MEN1 (0.64) MEN1MAPTKMT2ATDP1CYP3A4
Troglitazone SCHEMBL3050513 0.99 MEN1 (0.63) MEN1MAPTKMT2ATDP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 42211 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026087695-A1 TREATMENT FOR METABOLIC DISORDER SAPREME TECHNOLOGIES B.V. (NL) 2026-04-30 WO claimed
US-20260097039-A1 METHODS FOR TREATING A FATTY LIVER DISEASE MADRIGAL PHARMACEUTICALS INC (US) 2026-04-09 US claimed
US-20260069593-A1 METHODS FOR TREATING CANCER AMGEN INC (US) 2026-03-12 US claimed
US-20260048013-A1 PHARMACEUTICAL FORMULATION WITH IMPROVED SOLUBILITY AND BIOAVAILABILITY CONSEJO SUPERIOR INVESTIGACION (ES) 2026-02-19 US claimed
EP-4684799-A2 ANTIBODIES THAT DISRUPT THE INTERACTION OF GAL3 AND INSULIN RECEPTOR OR INTEGRINS AND METHODS OF USE THEREOF TrueBinding, Inc. (US) 2026-01-28 EP claimed
EP-4683679-A1 METHOD FOR DIAGNOSING AND TREATING NIS-EXPRESSING CARCINOMAS AND METASTASES NUSKE, Andreas (DE) 2026-01-28 EP claimed
EP-3452041-B1 COMPOSITIONS AND METHODS FOR ADMINISTERING PPAR-GAMMA-AGONISTS, SURFACTANT PEPTIDES AND PHOSPHOLIPIDS LOS ANGELES BIOMEDICAL RES INST HARBOR UCLA MEDICAL CT (US) 2026-01-14 EP claimed
US-12522805-B2 Method for obtaining cell spheroids D.I.V.A EXPERTISE (FR) 2026-01-13 US claimed
US-20250360215-A1 PHARMACEUTICAL COMBINATIONS AND METHODS FOR PREVENTING OR TREATING NEURODEGENERATIVE DISEASES YUH CHIOU HWA (US) 2025-11-27 US claimed
US-20250352528-A1 TOPICAL ROSIGLITAZONE FOR RADIATION-INDUCED SKIN INJURY BRIGHAM & WOMENS HOSPITAL INC (US) 2025-11-20 US claimed
US-5457109-A Use of thiazolidinedione derivatives and related antihyperglycemic agents in the treatment of disease states at risk for progressing to noninsulin-dependent diabetes mellitus WARNER-LAMBERT COMPANY (US) 1995-10-10 US claimed
CN-2207197-Y Heating medicinal band for diabetes XING GUANGMING (CN) 1995-09-13 CN claimed
WO-1995007694-A1 USE OF THIAZOLIDINEDIONES TO PREVENT OR DELAY ONSET OF NIDDM SANKYO COMPANY, LIMITED (JP) 1995-03-23 WO claimed
WO-1995007697-A2 USE OF THIAZOLIDINEDIONE DERIVATIVES AND RELATED ANTIHYPERGLYCEMIC AGENTS IN THE TREATMENT OF DISEASE STATES AT RISK FOR PROGRESSING TO NONINSULIN-DEPENDENT DIABETES MELLITUS WARNER-LAMBERT COMPANY (US) 1995-03-23 WO claimed
EP-0439321-B1 Thiazolidine derivatives having anti-hypertensive activity and their therapeutic use SANKYO CO (JP) 1995-03-15 EP claimed
EP-0617612-A1 A PROCESS FOR THE PREPARATION OF A SOLID DISPERSION. WARNER LAMBERT CO (US) 1994-10-05 EP claimed
WO-1993011749-A1 A PROCESS FOR THE PREPARATION OF A SOLID DISPERSION WARNER-LAMBERT COMPANY (US) 1993-06-24 WO claimed
EP-0139421-B1 THIAZOLIDINE DERIVATIVES, THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM SANKYO COMPANY LIMITED (JP) 1988-04-27 EP claimed
US-4572912-A Thiazolidine derivatives, their preparation and compositions containing them SANKYO COMPANY LIMITED (JP) 1986-02-25 US claimed
EP-0139421-A1 Thiazolidine derivatives, their preparation and compositions containing them SANKYO COMPANY LIMITED (JP) 1985-05-02 EP claimed