SCHEMBL4959062

SCHEMBL4959062

CN1CCN(c2ccnc3[nH]c4ccc(CCS(=O)(=O)c5ccccc5)cc4c23)CC1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 19/20 0.56
CHRM2 P08172 1/20 0.45
HTR1A P08908 1/20 0.45
ADRA2A P08913 1/20 0.45
CHRM1 P11229 1/20 0.45
DRD1 P21728 1/20 0.45
SLC6A2 P23975 1/20 0.45
HTR1B P28222 1/20 0.45
OPRM1 P35372 1/20 0.45
SLC6A3 Q01959 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14594930 0.91 ALK (0.58) ALK
SCHEMBL14594956 0.87 ALK (0.55) ALK
SCHEMBL14594934 0.81 ALK (0.47) ALK
SCHEMBL14626816 0.80 ALK (0.46) ALKHTR1AHTR1B
SCHEMBL14594932 0.80 ALK (0.51) ALK
SCHEMBL14594931 0.79 ALK (0.52) ALK
SCHEMBL14594933 0.79 ERBB2 (0.47) ALK
SCHEMBL14594959 0.79 ALK (0.45) ALK
SCHEMBL4962614 0.79 CHRM2 (0.40) ALKCHRM2HTR1AADRA2ACHRM1
SCHEMBL14594938 0.79 ALK (0.51) ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896472-A1 ALPHA-CARBOLINES AS CDK-1 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2008-03-12 EP disclosed
WO-2006131552-A1 ALPHA-CARBOLINES AS CDK-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-12-14 WO disclosed