SCHEMBL4962191

SCHEMBL4962191

Cc1ncc(-c2nc(Nc3ccc(C(=O)N(C)CCO)cc3)ncc2F)n1C1CCOCC1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 16/20 0.54
KCNH2 Q12809 7/20 0.54
CDK1 P06493 6/20 0.48
JAK2 O60674 2/20 0.43
JAK1 P23458 1/20 0.43
JAK3 P52333 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4250246 0.99 CDK2 (0.53) CDK2KCNH2CDK1JAK2JAK1
Hydrochloric Acid SCHEMBL4254788 0.90 CDK2 (0.51) CDK2KCNH2CDK1JAK2JAK1
Hydrochloric Acid SCHEMBL4246663 0.90 CDK2 (0.50) CDK2KCNH2CDK1JAK2JAK1
SCHEMBL13879011 0.88 CDK2 (0.54) CDK2KCNH2CDK1JAK2JAK1
Hydrochloric Acid SCHEMBL4247697 0.87 CDK2 (0.53) CDK2KCNH2CDK1JAK2JAK1
SCHEMBL13879010 0.86 CDK2 (0.54) CDK2KCNH2CDK1JAK2JAK1
SCHEMBL4243943 0.85 CDK2 (0.53) CDK2KCNH2CDK1JAK2JAK1
Hydrochloric Acid SCHEMBL4249706 0.85 CDK2 (0.53) CDK2KCNH2CDK1JAK2JAK1
Hydrochloric Acid SCHEMBL4250789 0.84 CDK2 (0.56) CDK2KCNH2CDK1JAK2JAK1
Lithium Ion SCHEMBL4243939 0.84 CDK2 (0.52) CDK2KCNH2CDK1JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945628-A1 NEW PYRIMIDINE DERIVATIVES AND THEIR USE IN THERAPY AS WELL AS THE USE OF PYRIMIDINE DERIVATIVES IN THE MANUFACTURE OF A MEDICAMENT FOR PREVENTION AND/OR TREATMENT OF ALZHEIMER'S DISEASE AstraZeneca AB (SE) 2008-07-23 EP claimed
WO-2007040440-A1 NEW PYRIMIDINE DERIVATIVES AND THEIR USE IN THERAPY AS WELL AS THE USE OF PYRIMIDINE DERIVATIVES IN THE MANUFACTURE OF A MEDICAMENT FOR PREVENTION AND/OR TREATMENT OF ALZHEIMER’S DISEASE ASTRAZENECA AB (SE) 2007-04-12 WO claimed