SCHEMBL4964392

SCHEMBL4964392

CCCNC(=O)C1CCCN1P(N)(=O)N1CCC[C@H](N)C1=O

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 5/20 0.44
NPSR1 Q6W5P4 1/20 0.35
GAA P10253 1/20 0.35
LCK P06239 2/20 0.35
LMNA P02545 1/20 0.34
FKBP1A P62942 4/20 0.34
MMP9 P14780 2/20 0.34
MMP3 P08254 1/20 0.34
PRCP P42785 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967075 0.80 DPP4 (0.49) DPP4
SCHEMBL4968943 0.75 DPP4 (0.51) DPP4LMNAKDM4E
SCHEMBL4965964 0.73 DPP4 (0.49) DPP4LMNA
SCHEMBL4965323 0.73 DPP4 (0.46) DPP4LMNA
SCHEMBL4968360 0.73 DPP4 (0.57) DPP4LMNA
SCHEMBL4964499 0.72 DPP4 (0.47) DPP4LMNA
SCHEMBL4964998 0.72 DPP4 (0.47) DPP4LCKLMNA
SCHEMBL4966271 0.72 DPP4 (0.48) DPP4LMNA
SCHEMBL4968301 0.71 DPP4 (0.46) DPP4KDM4EHPGD
SCHEMBL4965052 0.71 DPP4 (0.46) DPP4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1489088-B1 NOVEL ALPHA-AMINO-N-(DIAMINOPHOSPHINYL)LACTAM DERIVATIVE NIPPON KAYAKU KK (JP) 2008-08-13 EP disclosed
US-7348318-B2 α-Amino-N-(diaminophosphinyl)lactam derivatives NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2008-03-25 US disclosed
US-20050164989-A1 Novel $g(a)-amino-n-(diaminophosphinyl) lactam derivative NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2005-07-28 US disclosed
EP-1489088-A1 NOVEL ALPHA-AMINO-N-(DIAMINOPHOSPHINYL)LACTAM DERIVATIVE Nippon Kayaku Kabushiki Kaisha (JP) 2004-12-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050164989-A1 Novel $g(a)-amino-n-(diaminophosphinyl) lactam derivative DNPEP, PEPD, ANPEP DPP4 8/4885NPSR1 3444/4885GAA 43/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.