SCHEMBL4964892

SCHEMBL4964892

CCN(CC)C(=O)c1cc2c(nc(C)n2C)c(O)c1CCC(=O)c1ccccc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
CASP1 P29466 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CTNNB1 P35222 2/20 0.34
WNT3A P56704 2/20 0.34
HCRTR1 O43613 10/20 0.34
HCRTR2 O43614 10/20 0.34
PDE5A O76074 1/20 0.33
CYP3A4 P08684 1/20 0.33
PDE4A P27815 1/20 0.33
PDE6C P51160 1/20 0.33
PDE7A Q13946 1/20 0.33
PDE11A Q9HCR9 1/20 0.33
PDE10A Q9Y233 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4963781 0.90 CTNNB1 (0.35) KDM4EALDH1A1GAAHPGDCASP1
SCHEMBL4735946 0.85 ELANE (0.40) TSHRMAPK1KDM4EALDH1A1GAA
SCHEMBL4962551 0.84 CTNNB1 (0.35) MAPK1ALDH1A1HPGDCTNNB1WNT3A
SCHEMBL4965054 0.83 HCRTR1 (0.32) HCRTR1HCRTR2
SCHEMBL4961356 0.82 HTT (0.43) TSHRALDH1A1LMNAMEN1KMT2A
SCHEMBL4738299 0.82 HTT (0.46) TSHRALDH1A1LMNAMEN1KMT2A
SCHEMBL4963749 0.81 GSK3B (0.35) KDM4EALDH1A1HSD17B10CTNNB1WNT3A
SCHEMBL4963521 0.80 NPC1 (0.42) ALDH1A1MEN1RAB9AKMT2ADRD4
SCHEMBL4964158 0.80 NPC1 (0.36) CTNNB1WNT3ACYP3A4MEN1RAB9A
SCHEMBL4964361 0.79 IDO1 (0.38) MAPK1CTNNB1WNT3ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904454-A2 PROCESS FOR THE PRODUCTION OF INTERMADIATES FOR THE PREPARATION OF TRICYCLIC BENZIMIDAZOLES Nycomed GmbH (DE) 2008-04-02 EP disclosed
WO-2006136552-A2 PROCESS FOR THE PRODUCTION OF INTERMADIATES FOR THE PREPARATION OF TRICYCLIC BENZIMIDAZOLES NYCOMED GMBH (DE) 2006-12-28 WO disclosed