SCHEMBL4965148

SCHEMBL4965148

CCOC(=O)c1cccc(N2CCC(CN3CCC(Oc4ccc(Cl)c(Cl)c4)CC3)CC2)c1

nearest known ligand 0.79

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 20/20 0.79
CCR3 P51677 20/20 0.79
KCNH2 Q12809 17/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4968615 0.90 HRH1 (0.78) HRH1CCR3KCNH2
SCHEMBL4967633 0.88 HRH1 (1.00) HRH1CCR3KCNH2
SCHEMBL4967350 0.86 HRH1 (0.59) HRH1CCR3KCNH2
SCHEMBL4965732 0.86 CCR3 (0.57) HRH1CCR3KCNH2
SCHEMBL5972573 0.84 HRH1 (0.73) HRH1CCR3KCNH2
SCHEMBL5972369 0.84 HRH1 (0.75) HRH1CCR3KCNH2
SCHEMBL5002422 0.81 HRH1 (1.00) HRH1CCR3KCNH2
SCHEMBL4967248 0.81 HRH1 (0.78) HRH1CCR3KCNH2
SCHEMBL18841136 0.81 HRH1 (1.00) HRH1CCR3KCNH2
SCHEMBL4967396 0.80 HRH1 (1.00) HRH1CCR3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1625114-B1 Piperidine derivatives for the the treatment of chemokine or H1 mediated diseases ASTRAZENECA AB (SE) 2008-08-27 EP disclosed
US-20060264463-A1 Chemical compounds MEDTECH CONVERGENCE FUND, L.P. 2006-11-23 US disclosed
EP-1625114-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2006-02-15 EP disclosed
WO-2004099144-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-11-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060264463-A1 Chemical compounds CCR3, CCR1, CCR4 HRH1 38/4885CCR3 1/4885KCNH2 4041/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.