SCHEMBL4965460

SCHEMBL4965460

CC=C(NC)C(=O)O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18811995 1.00
SCHEMBL4965456 1.00
SCHEMBL19780334 0.79
SCHEMBL12320166 0.77
SCHEMBL14625691 0.77
SCHEMBL19780741 0.77
SCHEMBL28858723 0.77 KDM4E (0.39)
SCHEMBL19487260 0.75
SCHEMBL14520485 0.75
SCHEMBL14945608 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106045983-A Preparing method of Afatinib 苏州富士莱医药股份有限公司 2016-10-26 CN claimed
CN-113825816-B Two-component adhesive composition, articles made therefrom, and method of making the same 陶氏环球技术有限责任公司 2023-11-24 CN disclosed
US-20220177753-A1 TWO-COMPONENT ADHESIVE COMPOSITIONS, ARTICLES PREPARED WITH SAME AND PREPARATION METHODS THEREOF DOW GLOBAL TECHNOLOGIES LLC (US) 2022-06-09 US disclosed
EP-3969530-A1 TWO-COMPONENT ADHESIVE COMPOSITIONS, ARTICLES PREPARED WITH SAME AND PREPARATION METHODS THEREOF Dow Global Technologies LLC (US) 2022-03-23 EP disclosed
CN-113825816-A Two-part adhesive composition, articles made therefrom, and method of making same 陶氏环球技术有限责任公司 2021-12-21 CN disclosed
WO-2020227963-A1 TWO-COMPONENT ADHESIVE COMPOSITIONS, ARTICLES PREPARED WITH SAME AND PREPARATION METHODS THEREOF DOW GLOBAL TECHNOLOGIES LLC (US) 2020-11-19 WO disclosed
CN-102713618-B Protein Kinase Complexes and Inhibitors CELGENE AVILOMICS RES INC 2015-07-15 CN disclosed
WO-2012123966-A1 PROCESS FOR THE PREPARATION OF 4 -SUBSTITUTED -1, 4-DIHYDROPYRIDINES ARCH PHARMALABS LIMITED (IN) 2012-09-20 WO disclosed
EP-1883630-A2 METHODS OF SYNTHESIZING 6-ALKYLAMINOQUINOLINE DERIVATIVES Wyeth (US) 2008-02-06 EP disclosed
EP-1368315-B1 METHOD FOR PREPARING AMLODIPINE HANMI PHARM IND CO LTD (KR) 2007-10-17 EP disclosed
EP-1089974-A1 PROCESS TO PREPARE DIHYDROPYRIDINE AND DERIVATIVES THEREOF Hoechst Celanese Corporation (US) 2001-04-11 EP disclosed
US-5977369-A Process to prepare dihydropyridine and derivatives thereof NAPP TECHNOLOGIES, INC. (US) 1999-11-02 US disclosed
US-5808084-A Process for the preparation of 1,4-dihydropyridinedicarboxylic esters PFIZER, INC. (US) 1998-09-15 US disclosed
WO-1997024326-A1 PROCESS TO PREPARE DIHYDROPYRIDINE AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1997-07-10 WO disclosed
EP-0395182-A1 Herbicidal compounds SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1990-10-31 EP disclosed
US-4722931-A MUSCLE RELAXANTS LABORATORIOS DELAGRANGE (ES) 1988-02-02 US disclosed
US-4038399-A 1,4-DIHYDROPYRIDINE CARBOXYLIC ACID ESTERS USEFUL AS CORONARY VESSEL DILATORS AND ANTI-HYPERTENSIVES BAYER AKTIENGESELLSCHAFT (DT) 1977-07-26 US disclosed
US-4031104-A ANTIHYPERTENSIVE AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1977-06-21 US disclosed
US-3996234-A CORONARY VESSEL DILATORS, HYPOTENSIVES BAYER AKTIENGESELLSCHAFT (DT) 1976-12-07 US disclosed
US-3974275-A 1,4-Dihydropyridine carboxylic acid esters useful as coronary vessel dilators and anti-hypertensives BAYER AKTIENGESELLSCHAFT (DT) 1976-08-10 US disclosed