SCHEMBL4967979

SCHEMBL4967979

CCc1ccc(Cc2cc(I)c(O[C@H]3CCOC3)cc2Br)cc1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 13/20 0.38
PDE4A P27815 6/20 0.38
PDE4B Q07343 6/20 0.38
PDE4C Q08493 6/20 0.38
SLC5A2 P31639 6/20 0.35
SLC5A1 P13866 3/20 0.35
CHEK1 O14757 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967985 1.00 PDE4D (0.38) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL14116528 1.00 PDE4D (0.38) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL4966210 0.86 KMT2A (0.41) SLC5A2SLC5A1
SCHEMBL4966844 0.82 PDE4D (0.45) PDE4DPDE4APDE4BPDE4C
SCHEMBL4967088 0.82 PDE4D (0.45) PDE4DPDE4APDE4BPDE4C
SCHEMBL4967734 0.80 PDE4D (0.38) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL4968649 0.80 PDE4D (0.38) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL4967723 0.80 PDE4D (0.38) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL4966730 0.78 IKBKE (0.36) PDE4DPDE4APDE4BPDE4CSLC5A2
SCHEMBL4966718 0.78 IKBKE (0.36) PDE4DPDE4APDE4BPDE4CSLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed