SCHEMBL4968231

SCHEMBL4968231

NS(=O)(=O)c1ccc(-c2ccnc3[nH]ccc23)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 13/20 1.00
CHUK O15111 12/20 1.00
ROCK1 Q13464 2/20 0.67
NEK1 Q96PY6 6/20 0.66
PIK3C3 Q8NEB9 1/20 0.64
DAPK3 O43293 1/20 0.60
JAK2 O60674 1/20 0.60
PRKD3 O94806 1/20 0.60
MAP4K4 O95819 1/20 0.60
PAK4 O96013 1/20 0.60
CSF1R P07333 1/20 0.60
RET P07949 1/20 0.60
IGF1R P08069 1/20 0.60
FGFR1 P11362 1/20 0.60
PRKACA P17612 1/20 0.60
FLT1 P17948 1/20 0.60
LTK P29376 1/20 0.60
GRK5 P34947 1/20 0.60
KDR P35968 1/20 0.60
MAP2K2 P36507 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4792437 0.85 IKBKB (0.74) IKBKBCHUKROCK1NEK1PIK3C3
SCHEMBL12127248 0.83 IKBKB (1.00) IKBKBCHUKROCK1NEK1PIK3C3
SCHEMBL24805260 0.83 IKBKB (0.76) IKBKBCHUKROCK1NEK1PIK3C3
SCHEMBL24804168 0.80 IKBKB (0.66) IKBKBCHUKROCK1NEK1PIK3C3
SCHEMBL4792517 0.80 IKBKB (0.70) IKBKBCHUKROCK1NEK1DAPK3
SCHEMBL4968595 0.79 IKBKB (1.00) IKBKBCHUKROCK1NEK1PIK3C3
SCHEMBL30009321 0.77 IKBKB (0.66) IKBKBCHUKROCK1NEK1PIK3C3
SCHEMBL30009843 0.77 IKBKB (0.70) IKBKBCHUKROCK1NEK1PIK3C3
SCHEMBL30009837 0.77 IKBKB (0.66) IKBKBCHUKROCK1NEK1PIK3C3
SCHEMBL30009257 0.77 IKBKB (0.66) IKBKBCHUKROCK1NEK1PIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1962851-A2 COMPOUNDS SmithKline Beecham Corporation (US) 2008-09-03 EP disclosed
WO-2007076320-A2 COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed