SCHEMBL4972186

SCHEMBL4972186

CC(C)(C)N1CCC[C@H](Oc2cc(Cl)nc(N3CCOCC3)n2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.38
MEN1 O00255 2/20 0.38
PDE10A Q9Y233 2/20 0.37
RAF1 P04049 1/20 0.36
BRAF P15056 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.34
MAPT P10636 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PIK3CA P42336 2/20 0.34
PIK3R1 P27986 1/20 0.34
ACACB O00763 2/20 0.33
HTT P42858 2/20 0.33
CYP1A2 P05177 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17407919 0.84 PDE10A (0.43) KMT2AMEN1PDE10ARAF1BRAF
SCHEMBL2815435 0.82 PIK3CD (0.43) SMN1; SMN2PIK3CAPIK3R1
SCHEMBL2816228 0.82 PIK3CD (0.43) SMN1; SMN2PIK3CAPIK3R1
SCHEMBL2815436 0.82 PIK3CD (0.43) SMN1; SMN2PIK3CAPIK3R1
SCHEMBL4975886 0.81 EGLN1 (0.37) KMT2AMEN1PDE10ARAF1BRAF
SCHEMBL2815691 0.80 PDE10A (0.46) KMT2AMEN1PDE10ARAF1BRAF
SCHEMBL2813072 0.78 PIK3CD (0.48) PIK3CAPIK3R1
SCHEMBL2813469 0.78 PIK3CD (0.48) PIK3CAPIK3R1
SCHEMBL2813070 0.78 PIK3CD (0.48) PIK3CAPIK3R1
SCHEMBL2815645 0.77 JAK3 (0.44) KMT2AMEN1PDE10ARAF1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984350-A1 PYRIMIDINE DERIVATIVES USED AS PI-3 KINASE INHIBITORS Novartis AG (CH) 2008-10-29 EP disclosed
WO-2007084786-A1 PYRIMIDINE DERIVATIVES USED AS PI-3 KINASE INHIBITORS NOVARTIS AG (CH) 2007-07-26 WO disclosed