SCHEMBL4975648

SCHEMBL4975648

O=C(O)c1nnc(N2CCN(C(=O)CCN3CCCC3)CC2)nc1NCc1ccc(Cl)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 9/20 0.44
HTR1A P08908 6/20 0.42
HTR7 P34969 5/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
EPHX2 P34913 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4209221 0.89 CCR4 (0.42) CCR4HTR1AHTR7ALDH1A1MAPT
SCHEMBL4201714 0.83 EPHX2 (0.43) CCR4ALDH1A1EPHX2
SCHEMBL4205431 0.80 NPSR1 (0.43) CCR4ALDH1A1MAPTEPHX2
SCHEMBL13780306 0.76 NPSR1 (0.43) CCR4ALDH1A1MAPTTSHR
SCHEMBL4201718 0.75 KDM4E (0.40) CCR4ALDH1A1EPHX2
SCHEMBL13780107 0.74 EPHX2 (0.51) CCR4EPHX2
SCHEMBL13780154 0.74 EPHX2 (0.52) CCR4EPHX2
SCHEMBL13780152 0.74 EPHX2 (0.52) CCR4EPHX2
SCHEMBL13780307 0.73 CCR4 (0.44) CCR4EPHX2
SCHEMBL4216360 0.72 CCR4 (0.43) CCR4ALDH1A1MAPTEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1970373-A1 ALICYCLIC HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2008-09-17 EP disclosed