SCHEMBL4977205

SCHEMBL4977205

CC1CN(C(CO)c2cccnc2)CCN1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.45
SLC6A4 P31645 2/20 0.45
SLC6A3 Q01959 1/20 0.45
CACNA2D1 P54289 2/20 0.44
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
KCNA5 P22460 1/20 0.39
KCNH2 Q12809 1/20 0.39
SLC1A3 P43003 1/20 0.39
SLC1A2 P43004 1/20 0.39
SLC1A1 P43005 1/20 0.39
TP53 P04637 4/20 0.38
LMNA P02545 4/20 0.37
MAPT P10636 2/20 0.37
HSP90AA1 P07900 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4104611 1.00 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3CACNA2D1ALDH1A1
SCHEMBL4105919 1.00 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3CACNA2D1ALDH1A1
SCHEMBL4099505 0.84 OPRL1 (0.47) SLC6A2SLC6A4SLC6A3HRH3KCNH2
SCHEMBL4099664 0.84 OPRL1 (0.47) SLC6A2SLC6A4SLC6A3HRH3KCNH2
SCHEMBL4097078 0.76 TP53 (0.44) ALDH1A1KDM4EHSD17B10SLC1A2TP53
SCHEMBL4106918 0.76 TP53 (0.44) ALDH1A1KDM4EHSD17B10SLC1A2TP53
SCHEMBL14095780 0.70 SLC6A4 (0.52) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL20818025 0.70 SLC6A4 (0.63) SLC6A2SLC6A4SLC6A3ALDH1A1KDM4E
SCHEMBL13750181 0.70 HRH3 (0.47) SLC6A2SLC6A4SLC6A3CACNA2D1HRH3
SCHEMBL13749435 0.70 HRH3 (0.47) SLC6A2SLC6A4SLC6A3CACNA2D1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134036-A1 ALPHA-SUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-α]PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed