SCHEMBL4981087

SCHEMBL4981087

CCN(CC)c1ncc(N(CC)S(=O)(=O)c2ccccc2Cl)c(NC(Cc2ccc(OC(=O)N(C)C)cc2)C(=O)O)n1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.63
ITGA4 P13612 20/20 0.63
ITGB7 P26010 14/20 0.61
ITGAV P06756 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2769314 0.89 ITGB1 (0.60) ITGB1ITGA4ITGB7ITGAV
SCHEMBL2770988 0.88 ITGB1 (0.62) ITGB1ITGA4ITGB7ITGAV
SCHEMBL2773907 0.88 ITGB1 (0.61) ITGB1ITGA4ITGB7ITGAV
SCHEMBL2770133 0.86 ITGB1 (0.59) ITGB1ITGA4ITGB7ITGAV
SCHEMBL2769577 0.85 ITGB1 (0.69) ITGB1ITGA4ITGB7ITGAV
SCHEMBL2770949 0.85 ITGB1 (0.69) ITGB1ITGA4ITGB7ITGAV
SCHEMBL4981098 0.85 ITGB1 (0.62) ITGB1ITGA4ITGB7
SCHEMBL2770124 0.85 ITGB1 (0.64) ITGB1ITGA4ITGB7
SCHEMBL2769387 0.85 ITGB1 (0.61) ITGB1ITGA4ITGB7ITGAV
SCHEMBL4981105 0.84 ITGB1 (0.61) ITGB1ITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7335663-B2 Heteroaryl compounds which inhibit leukocyte adhesion mediated by α4 integrins ELAN PHARMACEUTICALS, INC. (US) 2008-02-26 US disclosed