SCHEMBL498942

SCHEMBL498942

CN(C[C@H](C[C@H]1CCCOC1)N(Cc1ccccc1)C(=O)O)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.38
SLC6A4 P31645 4/20 0.38
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
RORC P51449 1/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
ATM Q13315 1/20 0.34
KMT2A Q03164 2/20 0.33
HSD11B1 P28845 1/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
CACNA1B Q00975 1/20 0.33
MEN1 O00255 1/20 0.33
AKT1 P31749 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
NCOR2 Q9Y618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL499965 0.80 HTR2C (0.35) HTR2CSLC6A4ALDH1A1POLBHSD17B10
SCHEMBL8110118 0.79 SYK (0.46) KMT2ACTSLCTSBCTSSMEN1
SCHEMBL499680 0.78 ATM (0.38) RORCATMKMT2AMEN1ALDH1A1
SCHEMBL499442 0.76 HTR2C (0.31) HTR2CSLC6A4CTSLCTSBCTSS
SCHEMBL13242430 0.76 HTR2C (0.31) HTR2CSLC6A4CTSLCTSBCTSS
SCHEMBL2025474 0.75 SYK (0.43) KMT2ACTSLCTSBCTSSMEN1
SCHEMBL2025069 0.75 SYK (0.43) KMT2ACTSLCTSBCTSSMEN1
SCHEMBL2023544 0.75 SYK (0.43) KMT2ACTSLCTSBCTSSMEN1
SCHEMBL7992205 0.75 SYK (0.43) KMT2ACTSLCTSBCTSSMEN1
SCHEMBL2022224 0.75 SYK (0.43) KMT2ACTSLCTSBCTSSMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106221-B2 Renin inhibitors VITAE PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed