SCHEMBL500191

SCHEMBL500191

CC1C=CC=[C]N1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10811073 1.00
SCHEMBL906829 0.67
SCHEMBL312784 0.55
SCHEMBL6238732 0.55
SCHEMBL500342 0.54
SCHEMBL14452825 0.53
SCHEMBL14026153 0.53
SCHEMBL269336 0.53
SCHEMBL13270768 0.50
SCHEMBL22689369 0.50

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 122 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230174540-A1 3-(Carboxymethyl)-8-Amino-2-Oxo-1,3-Diaza-Spiro-[4.5]-Decane Derivatives GRUENENTHAL GMBH (DE) 2023-06-08 US disclosed
US-11572374-B2 N-cyano-7-azanorbornane derivatives and uses thereof AMGEN INC. (US) 2023-02-07 US disclosed
US-20210179627-A1 3-(Carboxymethyl)-8-Amino-2-Oxo-1,3-Diaza-Spiro-[4.5]-Decane Derivatives Grünenthal GmbH (DE) 2021-06-17 US disclosed
US-20200399280-A1 3-(Carboxymethyl)-8-Amino-2-Oxo-1,3-Diaza-Spiro-[4.5]-Decane Derivatives Grünenthal GmbH (DE) 2020-12-24 US disclosed
US-10807989-B2 3-(carboxymethyl)-8-amino-2-oxo-1,3-diaza-spiro-[4.5]-decane derivatives Grünenthal GmbH (DE) 2020-10-20 US disclosed
US-20190106430-A1 3-(CARBOXYMETHYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES Grünenthal GmbH (DE) 2019-04-11 US disclosed
US-20180282341-A1 3-(CARBOXYMETHYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES GRUENENTHAL GMBH (DE) 2018-10-04 US disclosed
US-9756858-B2 Insecticides SYNGENTA PARTICIPATIONS AG (CH) 2017-09-12 US disclosed
US-20160219879-A1 FUNGICIDAL COMPOSITIONS SYNGENTA PARTICIPATIONS AG (CH) 2016-08-04 US disclosed
US-9403845-B2 Pesticidally active pyridyl- and pyrimidyl- substituted pyrazole derivatives SYNGENTA PARTICIPATIONS AG (CH) 2016-08-02 US disclosed
WO-2006111341-A1 CYANO ANTHRANILAMIDE INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2006-10-26 WO disclosed
US-20060135517-A1 Imidazolopyridines and methods of making and using the same BIOGEN IDEC MA INC. 2006-06-22 US disclosed
WO-2006040113-A2 HETEROCYCLIC DIAMIDE INSECTICIDAL AGENTS SYNGENTA PARTICIPATIONS AG (CH) 2006-04-20 WO disclosed
WO-2006032462-A1 NOVEL INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2006-03-30 WO disclosed
US-20060052247-A1 Novel herbicides SYNGENTA CROP PROTECTION, INC. 2006-03-09 US disclosed
WO-2006024523-A1 PHTHALAMIDE DERIVATIVES FOR USE AS INSECTICIDES SYNGENTA PARTICIPATION AG (CH) 2006-03-09 WO disclosed
CN-1732166-A Novel herbicides SYNGENTA PARTICIPATIONS AG (CH) 2006-02-08 CN disclosed
US-20050222197-A1 Novel pyrazolopyridine derivatives as pharmaceutical agents BEIGHT DOUGLAS W 2005-10-06 US disclosed
EP-1578747-A2 NOVEL HERBICIDES Syngenta Participations AG (CH) 2005-09-28 EP disclosed
WO-2004058712-A2 HERBICIDALLY ACTIVE NICOTINOYL DERIVATES SYNGENTA PARTICIPATIONS AG (CH) 2004-07-15 WO disclosed