SCHEMBL500361

SCHEMBL500361

Cc1ccc(Br)c(C(=O)O)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 1/20 0.61
MYC P01106 1/20 0.51
LCK P06239 1/20 0.47
FYN P06241 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ALDH1A1 P00352 2/20 0.46
NOTUM Q6P988 1/20 0.46
GFER P55789 1/20 0.45
MCL1 Q07820 1/20 0.44
KDM4E B2RXH2 1/20 0.44
HSD17B10 Q99714 2/20 0.44
METAP2 P50579 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
MAOB P27338 1/20 0.43
CA5A P35218 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrazine SCHEMBL28177325 0.94 CSNK2A1 (0.55) CSNK2A1MYCLCKFYNMEN1
SCHEMBL27992485 0.84 MAPT (0.49) CSNK2A1MYCMEN1KMT2AALDH1A1
SCHEMBL29775265 0.83 CSNK2A1 (0.55) CSNK2A1MYCLCKFYNMEN1
SCHEMBL30844550 0.83 F2R (0.47) CSNK2A1MYCMEN1KMT2AKDM4E
SCHEMBL211284 0.83 CSNK2A1 (0.55) CSNK2A1MYCLCKFYNMEN1
SCHEMBL136961 0.83 F2R (0.47) CSNK2A1MYCMEN1KMT2AKDM4E
SCHEMBL11731746 0.81 CSNK2A1 (0.44) CSNK2A1MYCMEN1KMT2AALDH1A1
SCHEMBL13254950 0.81 MAPT (0.46) CSNK2A1MYCMEN1KMT2AHDAC7
SCHEMBL3735051 0.81 CSNK2A1 (0.44) CSNK2A1MYCMEN1KMT2AALDH1A1
SCHEMBL31627797 0.79 CSNK2A1 (0.68) CSNK2A1MEN1KMT2AALDH1A1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 455 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118184679-A Photothermal agent and preparation method thereof, photothermal nanoparticle and preparation method thereof, insulating material and self-repairing method of insulating material 中国石油天然气股份有限公司 2024-06-14 CN claimed
EP-1797186-B1 EXPRESSION SYSTEM, COMPONENTS THEREOF AND METHODS OF USE NAT RES COUNCIL CANADA (CA) 2016-05-25 EP claimed
US-8728759-B2 Reverse cumate repressor mutant NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2014-05-20 US claimed
CN-103224482-A Isocoumarin compound, derivatives and synthesis method thereof UNIV SHANGHAI JIAOTONG 2013-07-31 CN claimed
US-8373005-B2 Process for the synthesis of ethers of aromatic acids E I DU PONT DE NEMOURS AND COMPANY (US) 2013-02-12 US claimed
US-8252556-B2 Reverse cumate repressor mutant NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2012-08-28 US claimed
EP-2473469-A2 PROCESS FOR THE SYNTHESIS OF FLUORINATED ETHERS OF AROMATIC ACIDS E. I. du Pont de Nemours and Company (US) 2012-07-11 EP claimed
EP-2473470-A2 PROCESS FOR THE SYNTHESIS OF FLUORINATED ETHERS OF AROMATIC ACIDS E. I. du Pont de Nemours and Company (US) 2012-07-11 EP claimed
EP-2473468-A2 PROCESS FOR THE SYNTHESIS OF FLUORINATED ETHERS OF AROMATIC ACIDS E. I. du Pont de Nemours and Company (US) 2012-07-11 EP claimed
EP-2473471-A2 PROCESS FOR THE SYNTHESIS OF FLUORINATED ETHERS OF AROMATIC ACIDS E. I. du Pont de Nemours and Company (US) 2012-07-11 EP claimed
EP-1797186-A4 EXPRESSION SYSTEM, COMPONENTS THEREOF AND METHODS OF USE CA NAT RESEARCH COUNCIL (CA) 2008-11-12 EP claimed
WO-2008082510-A1 PROCESS FOR THE SYNTHESIS OF ETHERS OF AROMATIC ACIDS E.I. DU PONT DE NEMOURS AND COMPANY (US) 2008-07-10 WO claimed
WO-2008082551-A1 PROCESS FOR THE SYNTHESIS OF ETHERS OF AROMATIC ACIDS E.I. DU PONT DE NEMOURS AND COMPANY (US) 2008-07-10 WO claimed
WO-2008079225-A1 PROCESS FOR THE SYNTHESIS OF ETHERS OF AROMATIC ACIDS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2008-07-03 WO claimed
WO-2008079218-A1 PROCESS FOR THE SYNTHESIS OF ETHERS OF AROMATIC ACIDS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2008-07-03 WO claimed
EP-1797186-A1 EXPRESSION SYSTEM, COMPONENTS THEREOF AND METHODS OF USE NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2007-06-20 EP claimed
WO-2006037215-A1 EXPRESSION SYSTEM, COMPONENTS THEREOF AND METHODS OF USE NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2006-04-13 WO claimed
US-20040205834-A1 System for inducible expression in eukaryotic cells NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2004-10-14 US claimed
EP-1385946-A2 A SYSTEM FOR INDUCIBLE EXPRESSION IN EUKARYOTIC CELLS NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2004-02-04 EP claimed
WO-2002088346-A2 A SYSTEM FOR INDUCIBLE EXPRESSION IN EUKARYOTIC CELLS NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2002-11-07 WO claimed