SCHEMBL5014233

SCHEMBL5014233

CC(=O)OCc1cc2c(cn1)OCCN2C(=O)OCC(C)C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.37
GRM5 P41594 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 1/20 0.37
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
LMNA P02545 1/20 0.33
THRB P10828 1/20 0.33
NOTUM Q6P988 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP11B2 P19099 1/20 0.32
CYP3A4 P08684 1/20 0.32
SCN9A Q15858 1/20 0.32
SCN10A Q9Y5Y9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2937583 0.84 EGFR (0.41) MAPTGRM5ALDH1A1HTTPDE3B
SCHEMBL4428327 0.76 USP30 (0.40) MAPTGRM5ALDH1A1HTTPDE3B
SCHEMBL105404 0.73 CYP3A4 (0.47) MAPTALDH1A1HTTLMNAMEN1
SCHEMBL5744126 0.68 CTNNB1 (0.42) ALDH1A1NOTUMCYP3A4
SCHEMBL5140598 0.67 GRM5 (0.37) MAPTGRM5ALDH1A1HTTPDE3B
SCHEMBL4440734 0.67 HRH2 (0.42) ALDH1A1
SCHEMBL844057 0.63 CYP3A4 (0.39) ALDH1A1CYP3A4
SCHEMBL30412730 0.63 EGFR (0.43) MAPTGRM5ALDH1A1HTTPDE3B
SCHEMBL12405532 0.63 EGFR (0.43) MAPTGRM5THRBNOTUM
SCHEMBL12405526 0.63 EGFR (0.43) MAPTGRM5THRBNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001887-A1 PYRROLO-QUINOXALINONE DERIVATIVES AS ANTIBACTERIALS Glaxo Group Limited (GB) 2008-12-17 EP disclosed
WO-2007115947-A1 PYRROLO-QUINOXALINONE DERIVATIVES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2007-10-18 WO disclosed