SCHEMBL5016766

SCHEMBL5016766

CCS(=O)(=O)N1CCC(c2c[nH]c3c(C(N)=O)cc(-c4ccc(N5CCN(C(=O)OCC(C)C)CC5)nc4)cc23)CC1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 16/20 0.59
CHUK O15111 5/20 0.59
AURKA O14965 1/20 0.54
FLT3 P36888 1/20 0.54
CSNK1E P49674 1/20 0.54
BTK Q06187 1/20 0.54
GPR119 Q8TDV5 3/20 0.41
RET P07949 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL552028 0.89 IKBKB (0.60) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL551599 0.89 IKBKB (0.66) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL552981 0.87 IKBKB (0.70) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL551378 0.86 IKBKB (0.67) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL551885 0.85 IKBKB (0.68) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL551828 0.85 IKBKB (0.67) IKBKBCHUKAURKAFLT3CSNK1E
Trifluoroacetic Acid SCHEMBL551953 0.84 IKBKB (0.62) IKBKBCHUKAURKAFLT3CSNK1E
Trifluoroacetic Acid SCHEMBL553269 0.82 IKBKB (0.65) IKBKBCHUKAURKAFLT3CSNK1E
Trifluoroacetic Acid SCHEMBL552156 0.82 IKBKB (0.63) IKBKBCHUKAURKAFLT3CSNK1E
Trifluoroacetic Acid SCHEMBL551594 0.81 IKBKB (0.64) IKBKBCHUKAURKAFLT3CSNK1E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896014-A2 CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-03-12 EP disclosed
WO-2007005534-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-01-11 WO disclosed