SCHEMBL5016773

SCHEMBL5016773

CC(=O)SCCc1ccc2ccccc2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.53
PDE10A Q9Y233 2/20 0.46
RXFP1 Q9HBX9 3/20 0.44
PRNP P04156 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
MAPK10 P53779 1/20 0.44
GPBAR1 Q8TDU6 2/20 0.43
ALOX5 P09917 1/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
FFAR1 O14842 1/20 0.43
AKR1B1 P15121 1/20 0.43
LMNA P02545 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL728065 0.85 CYP1A2 (0.54) CYP1A2PDE10ARXFP1PRNPNPSR1
SCHEMBL14086502 0.80 PDE10A (0.50) CYP1A2PDE10ACYP2C19CYSLTR1
SCHEMBL5016772 0.78 PRNP (0.55) CYP1A2RXFP1PRNPNPSR1MAPK10
SCHEMBL27727433 0.78 CYP1A2 (0.57) CYP1A2PDE10AGPBAR1KDM4EMAPT
SCHEMBL2913941 0.76 PDE10A (0.61) CYP1A2PDE10ACYP2C19CYSLTR1
SCHEMBL4623799 0.76 CYP1A2 (0.68) CYP1A2PDE10ANPSR1GPBAR1ALOX5
SCHEMBL547194 0.75 FFAR1 (0.63) CYP1A2RXFP1PRNPNPSR1MAPK10
SCHEMBL29858122 0.74 HTT (0.55) CYP1A2HTTMEN1KMT2A
SCHEMBL10980763 0.74 CYP1A2 (0.53) CYP1A2PDE10AGPBAR1ALOX5MAPT
Acetic Acid SCHEMBL29172163 0.74 CYP1A2 (0.53) CYP1A2PDE10AGPBAR1ALOX5KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313751-B1 NEW MACROLIDES WITH ANTIBACTERIAL ACTIVITY BASILEA PHARMACEUTICA AG (CH) 2008-09-17 EP disclosed