SCHEMBL5016835

SCHEMBL5016835

CCCCn1c(=O)c2cc3c(cc2c2cnc4cc(OC)c(OC)cc4c21)OCO3

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 13/20 0.52
JAK2 O60674 3/20 0.47
JAK1 P23458 3/20 0.47
TYK2 P29597 3/20 0.47
JAK3 P52333 3/20 0.47
TNF P01375 2/20 0.43
LITAF Q99732 2/20 0.43
TDP2 O95551 1/20 0.42
NUAK1 O60285 1/20 0.40
NTRK1 P04629 1/20 0.40
FLT3 P36888 1/20 0.40
NUAK2 Q9H093 1/20 0.40
BMP2K Q9NSY1 1/20 0.40
LMNA P02545 1/20 0.40
THRB P10828 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4988592 0.98 TDP1 (0.52) TDP1JAK2JAK1TYK2JAK3
SCHEMBL19456961 0.88 TDP1 (0.54) TDP1JAK2JAK1TYK2JAK3
SCHEMBL4984289 0.88 TDP1 (0.51) TDP1JAK2JAK1TYK2JAK3
SCHEMBL241840 0.87 TDP1 (0.62) TDP1JAK2JAK1TYK2JAK3
SCHEMBL241835 0.87 TDP1 (0.53) TDP1JAK2JAK1TYK2JAK3
SCHEMBL241362 0.85 TDP1 (0.57) TDP1JAK2JAK1TYK2JAK3
Genz-644282 SCHEMBL29632787 0.85 TDP1 (0.52) TDP1JAK2JAK1TYK2JAK3
SCHEMBL29360706 0.85 TDP1 (0.69) TDP1JAK2JAK1TYK2JAK3
SCHEMBL241242 0.85 TDP1 (0.69) TDP1JAK2JAK1TYK2JAK3
Genz-644282 SCHEMBL241696 0.85 TDP1 (0.52) TDP1JAK2JAK1TYK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453812-B1 CYTOTOXIC AGENTS UNIV RUTGERS (US) 2008-08-20 EP disclosed