SCHEMBL5017145

SCHEMBL5017145

O=c1[nH]ccc2cc(CCO)c3ccc(-c4ccc(CN5CCOCC5)cc4)cc3c12

nearest known ligand 0.83

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 17/20 0.83
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ATM Q13315 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43
JAK2 O60674 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5017722 0.94 CHEK1 (0.80) CHEK1NPC1RAB9AATMHRH3
SCHEMBL4287873 0.92 CHEK1 (0.79) CHEK1NPC1RAB9AATMHRH3
SCHEMBL13659635 0.91 CHEK1 (0.84) CHEK1NPC1RAB9AATMHRH3
SCHEMBL4293965 0.91 CHEK1 (1.00) CHEK1NPC1RAB9AATMHRH3
SCHEMBL4292384 0.90 CHEK1 (0.82) CHEK1NPC1RAB9AATMHRH3
SCHEMBL4287654 0.89 CHEK1 (0.79) CHEK1NPC1RAB9AATMHRH3
SCHEMBL4292566 0.88 CHEK1 (0.71) CHEK1NPC1RAB9AATMHRH3
SCHEMBL4287256 0.88 CHEK1 (0.78) CHEK1NPC1RAB9AATMHRH3
SCHEMBL4289999 0.86 CHEK1 (0.75) CHEK1NPC1RAB9AATMHRH3
SCHEMBL4287406 0.85 CHEK1 (0.68) CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904449-A2 INHIBITORS OF CHECKPOINT KINASES Merck & Co., Inc. (US) 2008-04-02 EP claimed
WO-2007008502-A2 INHIBITORS OF CHECKPOINT KINASES MERCK & CO., INC. (US) 2007-01-18 WO claimed
EP-1904449-A2 INHIBITORS OF CHECKPOINT KINASES Merck & Co., Inc. (US) 2008-04-02 EP disclosed
WO-2007008502-A2 INHIBITORS OF CHECKPOINT KINASES MERCK & CO., INC. (US) 2007-01-18 WO disclosed