SCHEMBL5019540

SCHEMBL5019540

C[C@H](Nc1ncnc2cccnc12)c1cc2cccc(-c3cnn(C)c3)c2cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.44
ERBB2 P04626 2/20 0.44
ERBB4 Q15303 2/20 0.44
IRAK1 P51617 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
CREBBP Q92793 3/20 0.39
PIK3CD O00329 2/20 0.39
PIK3R2 O00459 1/20 0.39
PDPK1 O15530 1/20 0.39
RPS6KB1 P23443 1/20 0.39
AURKB Q96GD4 1/20 0.38
PIK3CG P48736 4/20 0.38
TTK P33981 4/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
PDE2A O00408 1/20 0.36
CHRM2 P08172 1/20 0.36
MET P08581 1/20 0.36
PDE4A P27815 1/20 0.36
PDE1A P54750 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4569488 0.82 PIK3CG (0.39) EGFRERBB2ERBB4IRAK1IRAK4
SCHEMBL14649370 0.79 PIK3CG (0.54) EGFRERBB2ERBB4IRAK1IRAK4
SCHEMBL4569401 0.79 PIK3CG (0.37) EGFRERBB2ERBB4IRAK1IRAK4
SCHEMBL4569410 0.79 IRAK4 (0.41) EGFRERBB2ERBB4IRAK1IRAK4
SCHEMBL4569435 0.78 PIK3CG (0.39) EGFRERBB2ERBB4PIK3CDPIK3R2
SCHEMBL4569411 0.78 PIK3CG (0.39) EGFRERBB2ERBB4IRAK1IRAK4
SCHEMBL14649241 0.77 PIK3CG (0.64) EGFRERBB2ERBB4PIK3CDPIK3R2
SCHEMBL14649174 0.77 PIK3CG (0.64) PIK3CDPIK3R2PIK3CGPDE3A
SCHEMBL4569447 0.77 PIK3CG (0.44) EGFRERBB2ERBB4IRAK4PIK3CD
SCHEMBL14667235 0.74 PIK3CG (0.59) PIK3CDPIK3R2PIK3CGPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064973-A2 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed