SCHEMBL5020123

SCHEMBL5020123

CCOC(=O)CNC(=O)[C@@H](N)Cc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPID Q08752 2/20 0.58
OPRK1 P41145 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
ABCC3 O15438 1/20 0.53
NR1I2 O75469 1/20 0.53
ABCB11 O95342 1/20 0.53
NR3C1 P04150 1/20 0.53
RARG P13631 1/20 0.53
CNR1 P21554 1/20 0.53
NR1H2 P55055 1/20 0.53
PPARA Q07869 1/20 0.53
NR1H3 Q13133 1/20 0.53
NR1I3 Q14994 1/20 0.53
MMP8 P22894 1/20 0.51
ALPI P09923 1/20 0.49
PKM P14618 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL11019745 0.99 PPID (0.57) PPIDOPRK1CYP1A2CYP3A4CYP2D6
Bromide SCHEMBL10788649 0.99 PPID (0.57) PPIDOPRK1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL10344243 0.99 PPID (0.57) PPIDOPRK1CYP1A2CYP3A4CYP2D6
SCHEMBL29007088 0.95 PPID (0.53) PPIDOPRK1CYP1A2CYP3A4CYP2D6
SCHEMBL29007089 0.95 PPID (0.53) PPIDOPRK1CYP1A2CYP3A4CYP2D6
SCHEMBL22539312 0.87 CYP1A2 (0.64) OPRK1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL7635307 0.87 SLC7A5 (0.53) OPRK1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6162382 0.87 SLC7A5 (0.53) OPRK1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL31303644 0.87 CYP3A4 (0.49) PPIDOPRK1CYP1A2CYP3A4CYP2D6
SCHEMBL24754621 0.86 PPID (0.47) PPIDOPRK1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012065102-A2 S-T-BUTYL PROTECTED CYSTEINE DI-PEPTIDE ANALOGS AND RELATED COMPOUNDS PROMENTIS PHARMACEUTICALS, INC. (US) 2012-05-18 WO disclosed
US-3984417-A Method of producing active amino acid esters AJINOMOTO CO., INC. (JA) 1976-10-05 US disclosed
US-3933783-A Formation of peptide bonds in the presence of isonitriles AJINOMOTO CO., INC. (JA) 1976-01-20 US disclosed