SCHEMBL5020929

SCHEMBL5020929

CNc1nc(Nc2cn(C(F)F)nc2C)ncc1N

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 20/20 0.58
CYP1A2 P05177 6/20 0.58
TTK P33981 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5021244 0.89 LRRK2 (0.69) LRRK2CYP1A2TTK
SCHEMBL4562047 0.85 LRRK2 (0.58) LRRK2CYP1A2TTK
SCHEMBL4559379 0.83 LRRK2 (0.83) LRRK2CYP1A2TTK
SCHEMBL4540863 0.82 LRRK2 (0.55) LRRK2CYP1A2TTK
SCHEMBL5021245 0.79 LRRK2 (0.69) LRRK2CYP1A2TTK
SCHEMBL10286422 0.78 LRRK2 (0.61) LRRK2CYP1A2TTK
SCHEMBL5021224 0.77 LRRK2 (0.57) LRRK2CYP1A2TTK
SCHEMBL5020930 0.77 LRRK2 (0.47) LRRK2CYP1A2TTK
SCHEMBL5021217 0.77 LRRK2 (0.47) LRRK2CYP1A2TTK
SCHEMBL5021213 0.77 LRRK2 (0.58) LRRK2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012062783-A1 PYRAZOLE AMINOPYRIMIDINE DERIVATIVES AS LRRK2 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-05-18 WO disclosed