SCHEMBL5021373

SCHEMBL5021373

CC(=O)CC1CCCc2cccnc21

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.41
CXCR4 P61073 10/20 0.40
CYP2D6 P10635 3/20 0.40
ADORA2A P29274 1/20 0.38
OPRL1 P41146 1/20 0.38
KCNH2 Q12809 1/20 0.38
CHRM3 P20309 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3311293 0.87 HDAC1 (0.46) HDAC1HDAC6PTGDR2CXCR4CYP2D6
SCHEMBL1698205 0.86 HDAC1 (0.40) HDAC1HDAC6PTGDR2CXCR4CYP2D6
SCHEMBL1698225 0.86 HDAC1 (0.40) HDAC1HDAC6PTGDR2CXCR4CYP2D6
SCHEMBL923694 0.83 PTGDR2 (0.44) HDAC1HDAC6PTGDR2CXCR4ADORA2A
SCHEMBL24858718 0.80 CYP2D6 (0.43) HDAC1HDAC6CXCR4CYP2D6
SCHEMBL3314390 0.80 HDAC1 (0.44) HDAC1HDAC6CXCR4CYP2D6
SCHEMBL21202393 0.80 CYP2D6 (0.43) HDAC1HDAC6CXCR4CYP2D6
SCHEMBL21275417 0.79 HDAC1 (0.42) HDAC1HDAC6CXCR4CYP2D6CHRM3
SCHEMBL2725023 0.79 HDAC1 (0.42) HDAC1HDAC6CXCR4CYP2D6CHRM3
SCHEMBL3950796 0.79 HDAC1 (0.43) HDAC1HDAC6CXCR4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120115893-A1 Substituted Bicyclic Carboxamide and Urea Compounds as Vanilloid Receptor Ligands GRUENENTHAL GMBH (DE) 2012-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120115893-A1 Substituted Bicyclic Carboxamide and Urea Compounds as Vanilloid Receptor Ligands TRPV1, CNR1, CNR2 HDAC1 606/4885HDAC6 704/4885PTGDR2 357/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.