SCHEMBL5021735

SCHEMBL5021735

O=C1N[C@H](c2cccnc2)[C@@H](c2ccc(F)cc2)O1

nearest known ligand 0.71

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 20/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5022138 0.88 GRM5 (0.55) GRM5
SCHEMBL5022139 0.88 GRM5 (0.55) GRM5
SCHEMBL5022091 0.86 GRM5 (0.71) GRM5
SCHEMBL13642274 0.86 GRM5 (0.71) GRM5
SCHEMBL4561532 0.84 GRM5 (1.00) GRM5
SCHEMBL13585577 0.84 GRM5 (1.00) GRM5
SCHEMBL4539727 0.80 GRM5 (0.67) GRM5
SCHEMBL16363427 0.80 GRM5 (0.60) GRM5
SCHEMBL16363933 0.80 GRM5 (0.62) GRM5
SCHEMBL5021968 0.79 GRM5 (0.73) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638022-B1 OXAZOLIDINONES AS MODULATORS OF MGLUR5 BRISTOL MYERS SQUIBB CO (US) 2014-12-24 EP disclosed
WO-2012064603-A1 OXAZOLIDINONES AS MODULATORS OF MGLUR5 BRISTOL-MYERS SQUIBB COMPANY (US) 2012-05-18 WO disclosed