SCHEMBL5029762

SCHEMBL5029762

CC(O)C(F)n1cnc2c(N)ncnc21

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.67
ADORA1 P30542 3/20 0.67
ADORA2B P29275 2/20 0.67
PI4KA P42356 1/20 0.67
PI4K2B Q8TCG2 1/20 0.67
PI4K2A Q9BTU6 1/20 0.67
PI4KB Q9UBF8 1/20 0.67
ADA P00813 4/20 0.57
PDE2A O00408 3/20 0.57
CYP3A4 P08684 2/20 0.57
PDE4A P27815 1/20 0.57
PDE4B Q07343 1/20 0.57
PDE4C Q08493 1/20 0.57
PDE4D Q08499 1/20 0.57
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
CYP1A2 P05177 1/20 0.57
ALOX15 P16050 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
HSD17B10 Q99714 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4813561 0.84 ADORA2A (0.75) ADORA2AADORA1ADORA2BPI4KAPI4K2B
Hydrochloric Acid SCHEMBL9193025 0.83 ADORA2A (0.73) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL754007 0.80 ADORA2A (1.00) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL28731072 0.80 ADORA2A (0.69) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL22474983 0.80 ADORA2A (0.69) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL24205121 0.79 ADORA2A (0.77) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL18521145 0.79 ADORA2A (0.77) ADORA2AADORA1ADORA2BPI4KAPI4K2B
Hydrochloric Acid SCHEMBL30881556 0.79 ADORA2A (0.96) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL19049967 0.78 ADORA2A (0.50) ADORA2AADORA1ADORA2BPI4KAPI4K2B
SCHEMBL8955888 0.78 ADORA2A (0.75) ADORA2AADORA1ADORA2BPI4KAPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134578-A2 SYNTHESIS OF OPTICALLY ACTIVE RADIO-LABELED REVERSE TRANSCRIPTASE INHIBITORS THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF (US) 2008-11-06 WO disclosed