SCHEMBL5035544

SCHEMBL5035544

CN(c1cccnc1)c1[c]cccn1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 3/20 0.47
GRM5 P41594 4/20 0.35
CHRNB2 P17787 3/20 0.35
CHRNA4 P43681 3/20 0.35
NOTUM Q6P988 1/20 0.35
CYP2A6 P11509 2/20 0.34
SYK P43405 1/20 0.33
KCNN4 O15554 1/20 0.33
CHRNA7 P36544 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27549059 0.77 KCNA5 (0.51) KCNA5GRM5CHRNB2CHRNA4NOTUM
SCHEMBL3409401 0.76 KCNA5 (0.49) KCNA5GRM5CHRNB2CHRNA4CYP2A6
Hydrochloric Acid SCHEMBL4024971 0.74 KCNA5 (0.47) KCNA5GRM5CHRNB2CHRNA4CYP2A6
SCHEMBL13443083 0.71 KCNA5 (0.47) KCNA5GRM5CHRNB2CHRNA4NOTUM
SCHEMBL10094607 0.71 KCNA5 (0.57) KCNA5GRM5CHRNB2CHRNA4NOTUM
SCHEMBL5075470 0.71 KCNA5 (0.50) KCNA5GRM5CHRNB2CHRNA4NOTUM
SCHEMBL1097763 0.70
SCHEMBL12919963 0.70 KCNA5 (0.46) KCNA5GRM5CHRNB2CHRNA4
SCHEMBL4770280 0.70 KCNA5 (0.40) KCNA5GRM5CHRNB2CHRNA4NOTUM
SCHEMBL29435745 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940406-A2 POTASSIUM CHANNEL INHIBITORS Merck and Co., Inc. (US) 2008-07-09 EP disclosed
WO-2007050348-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-05-03 WO disclosed