SCHEMBL5036060

SCHEMBL5036060

NC(=O)Oc1csc(N(C(=O)c2ccc(Cl)cc2Cl)c2ccc(Cl)cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.43
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
KMT2A Q03164 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAPT P10636 3/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
HPGD P15428 1/20 0.36
CASP3 P42574 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
KDM4E B2RXH2 2/20 0.35
PKM P14618 1/20 0.34
TSHR P16473 1/20 0.34
CASP1 P29466 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GABRA1 P14867 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5041330 0.87 CYP3A4 (0.44) CYP3A4CYP11B1CYP11B2KMT2ACYP1A2
SCHEMBL5032567 0.85 CYP3A4 (0.49) CYP3A4CYP11B1CYP11B2KMT2ACYP1A2
SCHEMBL5034868 0.83 CYP3A4 (0.45) CYP3A4KMT2AMAPTNPC1RAB9A
SCHEMBL5036077 0.82 CYP3A4 (0.42) CYP3A4CYP11B1CYP11B2KMT2ACYP1A2
SCHEMBL5034877 0.82 CYP3A4 (0.44) CYP3A4CYP11B1CYP11B2KMT2ACYP1A2
SCHEMBL5039110 0.82 CYP3A4 (0.42) CYP3A4CYP11B1CYP11B2KMT2ACYP1A2
SCHEMBL5041385 0.81 CYP3A4 (0.46) CYP3A4CYP11B1CYP11B2KMT2ACYP1A2
SCHEMBL5034908 0.81 CYP3A4 (0.43) CYP3A4CYP11B1CYP11B2KMT2ACYP1A2
SCHEMBL5035235 0.81 CYP3A4 (0.45) CYP3A4CYP11B1CYP11B2KMT2ACYP1A2
SCHEMBL5041312 0.81 CYP3A4 (0.40) CYP3A4CYP11B1CYP11B2KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694673-B1 THIAZOLE DERIVATES HOFFMANN LA ROCHE (CH) 2008-01-16 EP claimed