SCHEMBL5036183

SCHEMBL5036183

CN(C)S(=O)(=O)c1cccc(NC(=O)Oc2cnn3c(C(F)F)cc(-c4ccc(C(F)(F)F)cc4)nc23)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.52
KDM4E B2RXH2 3/20 0.52
HTT P42858 1/20 0.52
MAPK1 P28482 1/20 0.51
TP53 P04637 2/20 0.44
POLB P06746 1/20 0.44
LMNA P02545 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 3/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5034971 0.92 KDM4E (0.51) KMT2AKDM4EHTTMAPK1TP53
SCHEMBL5039150 0.92 KDM4E (0.54) KMT2AKDM4EHTTMAPK1TP53
SCHEMBL5035072 0.90 KDM4E (0.54) KMT2AKDM4EHTTMAPK1TP53
SCHEMBL5035253 0.90 MAPK1 (0.52) KMT2AKDM4EHTTMAPK1TP53
SCHEMBL5034992 0.90 MAPK1 (0.52) KMT2AKDM4EHTTMAPK1TP53
SCHEMBL5036473 0.90 KDM4E (0.44) KMT2AKDM4EHTTMAPK1POLB
SCHEMBL5035267 0.90 MAPK1 (0.48) KMT2AKDM4EHTTMAPK1TP53
SCHEMBL5032722 0.89 KDM4E (0.51) KMT2AKDM4EHTTMAPK1TP53
SCHEMBL5035008 0.89 KDM4E (0.51) KMT2AKDM4EHTTMAPK1TP53
SCHEMBL5035052 0.88 KDM4E (0.51) KMT2AKDM4EHTTMAPK1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed