SCHEMBL5037294

SCHEMBL5037294

O=C1C=CC2=C(CC=NC2=O)C1

nearest known ligand 0.39

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL277815 0.60
SCHEMBL1199564 0.58
SCHEMBL9847743 0.57 GSK3A (0.40) GSK3AGSK3B
SCHEMBL10790767 0.57 GSK3A (0.46) GSK3AGSK3B
SCHEMBL366153 0.56 GSK3A (0.71) GSK3AGSK3B
SCHEMBL353266 0.54 GSK3A (0.42) GSK3AGSK3B
SCHEMBL12505051 0.54 GSK3A (0.42) GSK3AGSK3B
SCHEMBL16093525 0.54
SCHEMBL14703233 0.52
SCHEMBL9527717 0.52 GSK3A (0.46) GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117730082-A Synthesis of substituted tricyclic amides and analogs thereof 爱彼特生物制药公司 2024-03-19 CN claimed
CN-117730082-A Synthesis of substituted tricyclic amides and analogs thereof 爱彼特生物制药公司 2024-03-19 CN disclosed
CN-115551864-A Substituted tricyclic amides, analogs thereof, and methods of using the same 爱彼特生物制药公司 2022-12-30 CN disclosed
CN-115087486-A Substituted bicyclic and tricyclic ureas and amides, analogs thereof, and methods of use thereof 爱彼特生物制药公司 2022-09-20 CN disclosed
EP-1667982-A4 ISOQUINOLINONE POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2008-08-13 EP disclosed
EP-1667982-A2 ISOQUINOLINONE POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2006-06-14 EP disclosed
WO-2005030791-A2 ISOQUINOLINONE POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2005-04-07 WO disclosed