SCHEMBL5039645

SCHEMBL5039645

O=c1ccc(-c2ccc(F)nc2)c[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.48
MAP4K4 O95819 1/20 0.47
PDGFRB P09619 1/20 0.46
PDGFRA P16234 1/20 0.46
CYP2A6 P11509 3/20 0.44
CYP2B6 P20813 3/20 0.44
CYP2E1 P05181 1/20 0.44
GRM5 P41594 1/20 0.42
DGAT1 O75907 1/20 0.40
SOAT1 P35610 1/20 0.40
KCNH2 Q12809 1/20 0.40
CYP11B2 P19099 1/20 0.38
MAPT P10636 5/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C19 P33261 2/20 0.38
JAK2 O60674 1/20 0.37
RET P07949 1/20 0.37
KDR P35968 1/20 0.37
GSK3A P49840 1/20 0.37
RPS6KA3 P51812 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26104326 0.77 CYP2A6 (0.64) CYP2A6CYP2B6CYP2E1GRM5CYP11B2
SCHEMBL23346571 0.76 PDGFRB (0.50) NPY5RMAP4K4PDGFRBPDGFRAGRM5
SCHEMBL26953398 0.76 MAP4K4 (0.48) NPY5RMAP4K4PDGFRBPDGFRAGRM5
SCHEMBL11161344 0.74 ERCC1 (0.53) NPY5RMAP4K4PDGFRBPDGFRAGRM5
SCHEMBL30279632 0.73 AKT2 (0.50) CYP2A6CYP2B6CYP2E1CYP11B2MAPT
SCHEMBL14783574 0.73 AKT2 (0.50) CYP2A6CYP2B6CYP2E1CYP11B2MAPT
SCHEMBL27422573 0.73 CYP2A6 (0.40) CYP2A6CYP2B6CYP2E1CYP11B2MAPT
SCHEMBL10843366 0.72 MAP4K4 (0.41) MAP4K4PDGFRBPDGFRAGRM5DGAT1
SCHEMBL13575357 0.71 AURKA (0.50) MAP4K4PDGFRBPDGFRACYP2A6GRM5
SCHEMBL11169629 0.70 TNKS2 (0.50) MAP4K4CLK4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871368-A2 DIHYDROPYRIDINE COMPOUNDS FOR NEURODEGENERATIVE DISEASES AND DEMENTIA Eisai Co., Ltd. (JP) 2008-01-02 EP disclosed
WO-2006107859-A2 DIHYDROPYRIDINE COMPOUNDS FOR NEURODEGENERATIVE DISEASES AND DEMENTIA EISAI CO., LTD. (JP) 2006-10-12 WO disclosed