SCHEMBL5041391

SCHEMBL5041391

NS(=O)(=O)c1cccc(NC(=O)Oc2cnn3c(C(F)F)cc(-c4ccc(C(F)(F)F)c(F)c4)nc23)c1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.48
KDM4E B2RXH2 3/20 0.48
HTT P42858 1/20 0.48
KMT2A Q03164 1/20 0.48
CA12 O43570 3/20 0.42
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
CA9 Q16790 3/20 0.42
TP53 P04637 2/20 0.42
POLB P06746 1/20 0.42
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5035331 0.93 KDM4E (0.49) MAPK1KDM4EHTTKMT2ATP53
SCHEMBL5036051 0.92 MAPK1 (0.49) MAPK1KDM4EHTTKMT2ACA12
SCHEMBL5036550 0.92 KDM4E (0.49) MAPK1KDM4EHTTKMT2ACA12
SCHEMBL5041451 0.91 MAPK1 (0.47) MAPK1KDM4EHTTKMT2ACA12
SCHEMBL5041375 0.90 HPGD (0.43) MAPK1KDM4EKMT2ACA12CA1
SCHEMBL5034992 0.89 MAPK1 (0.52) MAPK1KDM4EHTTKMT2ACA12
SCHEMBL5032681 0.89 KDM4E (0.47) MAPK1KDM4EHTTKMT2ACA12
SCHEMBL5048285 0.88 MAPK1 (0.58) MAPK1KDM4EHTTKMT2ACA12
SCHEMBL5034984 0.87 KDM4E (0.54) MAPK1KDM4EHTTKMT2ACA12
SCHEMBL5034903 0.86 MAPK1 (0.52) MAPK1KDM4EHTTKMT2ACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed