SCHEMBL5043150

SCHEMBL5043150

Nc1ccccc1NC(=O)c1ccc(N2CC3CCC(C2)N3C(=O)O)nc1

nearest known ligand 0.75

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 20/20 0.75
KCNH2 Q12809 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4533828 0.86 HDAC1 (1.00) HDAC1
SCHEMBL4538609 0.86 HDAC1 (1.00) HDAC1KCNH2
SCHEMBL4541782 0.81 HDAC1 (1.00) HDAC1KCNH2
SCHEMBL4541780 0.81 HDAC1 (1.00) HDAC1KCNH2
SCHEMBL4541792 0.81 HDAC1 (0.94) HDAC1
SCHEMBL4530382 0.80 HDAC1 (1.00) HDAC1
SCHEMBL8161162 0.80 HDAC1 (0.70) HDAC1KCNH2
SCHEMBL4526024 0.80 HDAC1 (1.00) HDAC1
SCHEMBL2410399 0.80 HDAC1 (0.65) HDAC1
SCHEMBL4540246 0.79 HDAC1 (0.83) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945028-A2 SUBSTITUTED NICOTINAMIDE COMPOUNDS Merck & Co., Inc. (US) 2008-07-23 EP disclosed
WO-2007055942-A2 SUBSTITUTED NICOTINAMIDE COMPOUNDS MERCK & CO., INC. (US) 2007-05-18 WO disclosed