SCHEMBL5046874

SCHEMBL5046874

CC(C)(C)OC(=O)n1c(-c2ccc(Cl)c3c2CNC3)cc2cc(Br)ccc21

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 1/20 0.41
CDK1 P06493 1/20 0.41
CCNB1 P14635 1/20 0.41
GSK3B P49841 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41
NR1H2 P55055 16/20 0.40
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40
NR1H3 Q13133 4/20 0.37
TTK P33981 1/20 0.36
ATR Q13535 1/20 0.36
ATRIP Q8WXE1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5049582 0.86 NR1H2 (0.47) NR1H2BRD4CREBBPNR1H3ATR
SCHEMBL3043890 0.76 BRD4 (0.38) NR1H2BRD4CREBBPNR1H3TTK
SCHEMBL5046843 0.75 NR1H2 (0.41) NR1H2BRD4CREBBPNR1H3ATR
SCHEMBL3044227 0.75 BRD4 (0.39) NR1H2BRD4CREBBPNR1H3ATR
SCHEMBL31694045 0.74 NR1H2 (0.59) NR1H2NR1H3
SCHEMBL3034386 0.74 BRD4 (0.51) NR1H2BRD4CREBBPNR1H3
SCHEMBL3047590 0.73 NR1H2 (0.45) NR1H2BRD4CREBBPNR1H3ATR
SCHEMBL3037160 0.73 ATR (0.40) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL21629674 0.73 NR1H2 (0.43) NR1H2NR1H3TTK
SCHEMBL3039340 0.73 BRD4 (0.37) NR1H2BRD4CREBBPATRATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed