SCHEMBL5047037

SCHEMBL5047037

Cc1cc(S(=O)(=O)Oc2ccc(-c3cc4cc(CN5CCCCC5)ccc4[nH]3)c3c2CNC3=O)c(C)s1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 16/20 0.43
AURKA O14965 3/20 0.40
KDR P35968 3/20 0.40
CDK7 P50613 3/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3050822 0.86 CHEK1 (0.45) CHEK1AURKAKDRCDK7
SCHEMBL3039315 0.86 CHEK1 (0.42) CHEK1AURKAKDRCDK7
SCHEMBL3039404 0.86 CHEK1 (0.47) CHEK1AURKAKDRCDK7
Hydrochloric Acid SCHEMBL3034106 0.86 CHEK1 (0.47) CHEK1AURKAKDRCDK7TSHR
SCHEMBL3040222 0.86 CHEK1 (0.48) CHEK1AURKAKDR
SCHEMBL3048839 0.85 AURKA (0.42) CHEK1AURKAKDR
SCHEMBL3043821 0.85 CHEK1 (0.41) CHEK1AURKAKDRCDK7
SCHEMBL3046134 0.85 CHEK1 (0.44) CHEK1AURKAKDRCDK7
SCHEMBL3048160 0.85 CHEK1 (0.45) CHEK1AURKAKDRCDK7
SCHEMBL3050852 0.85 CHEK1 (0.49) CHEK1AURKAKDRCDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed