SCHEMBL5047121

SCHEMBL5047121

Cc1c(OC(=O)NCC2CCCCC2)cc(-c2csc(-c3cnccn3)n2)n1CC1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.38
KLK1 P06870 1/20 0.38
CPT2 P23786 1/20 0.37
CPT1A P50416 1/20 0.37
CPT1B Q92523 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
PIM1 P11309 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
SCN9A Q15858 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
CNR2 P34972 1/20 0.31
F2RL3 Q96RI0 1/20 0.31
CDC7 O00311 1/20 0.31
DBF4 Q9UBU7 1/20 0.31
ACHE P22303 2/20 0.31
HTR4 Q13639 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5044141 0.86 KLKB1 (0.48) KLKB1KLK1CPT2CPT1ACPT1B
SCHEMBL5039914 0.82 CDC25A (0.45) KLKB1SMN1; SMN2ALDH1A1
SCHEMBL5039577 0.81 KLKB1 (0.42) KLKB1KLK1CPT2CPT1ACPT1B
SCHEMBL5043868 0.79 KLKB1 (0.46) KLKB1KLK1CPT2CPT1ACPT1B
SCHEMBL6069189 0.79 KLKB1 (0.46) KLKB1KLK1CPT2CPT1ACPT1B
SCHEMBL5039559 0.79 KLKB1 (0.46) KLKB1KLK1CPT2CPT1ACPT1B
SCHEMBL5045879 0.79 KLKB1 (0.44) KLKB1KLK1HDAC1HDAC8HDAC6
SCHEMBL5047187 0.78 HDAC3 (0.36) HDAC1HDAC6SMN1; SMN2ALDH1A1GAA
SCHEMBL5048938 0.78 KLKB1 (0.46) KLKB1KLK1CPT2CPT1ACPT1B
SCHEMBL5039321 0.78 KLKB1 (0.45) KLKB1KLK1CPT2CPT1ACPT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583762-B1 PYRROLYL-THIAZOLES AND THEIR USE AS CB 1 RECEPTOR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP claimed