SCHEMBL5048292

SCHEMBL5048292

COc1cc(-c2cc3cc(CN(C)C)ccc3n2C(=O)OC(C)(C)C)c2c(c1OS(=O)(=O)c1ccccc1C#N)CNC2=O

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 18/20 0.40
NR1H3 Q13133 3/20 0.35
JAK3 P52333 1/20 0.32
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3039557 0.90 NR1H2 (0.40) NR1H2NR1H3
SCHEMBL3037846 0.89 NR1H2 (0.35) NR1H2NR1H3JAK3BRD4CREBBP
SCHEMBL3044795 0.88 NR1H2 (0.35) NR1H2NR1H3JAK3BRD4CREBBP
SCHEMBL3045855 0.88 NR1H2 (0.42) NR1H2NR1H3BRD4CREBBP
SCHEMBL3049636 0.86 NR1H2 (0.32) NR1H2NR1H3JAK3
SCHEMBL3047406 0.84 NR1H2 (0.37) NR1H2NR1H3
SCHEMBL3049642 0.84 NR1H2 (0.37) NR1H2NR1H3JAK3BRD4CREBBP
SCHEMBL3048540 0.82 NR1H2 (0.34) NR1H2NR1H3
SCHEMBL3051211 0.82 NR1H2 (0.35) NR1H2NR1H3
SCHEMBL3037585 0.81 NR1H2 (0.34) NR1H2NR1H3BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed