SCHEMBL5048339

SCHEMBL5048339

CC(C)(C)OC(=O)n1c(-c2ccc(-c3ccco3)c3c2C(=O)NC3)cc2cc(CN3CCCCC3)ccc21

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EED O75530 1/20 0.36
NR1H2 P55055 12/20 0.35
TGFBR1 P36897 1/20 0.35
ATR Q13535 2/20 0.35
ATRIP Q8WXE1 2/20 0.35
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
NR1H3 Q13133 3/20 0.34
TBK1 Q9UHD2 1/20 0.32
PARP1 P09874 1/20 0.32
PIK3R1 P27986 1/20 0.32
PIK3CA P42336 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3042659 0.92 NR1H2 (0.36) EEDNR1H2ATRATRIPBRD4
SCHEMBL3033517 0.92 EED (0.34) EEDNR1H2TGFBR1ATRATRIP
SCHEMBL3046959 0.88 NR1H2 (0.41) NR1H2BRD4CREBBPNR1H3
SCHEMBL3049701 0.88 NR1H2 (0.37) NR1H2ATRATRIPBRD4CREBBP
SCHEMBL3039052 0.87 NR1H2 (0.37) NR1H2ATRATRIPBRD4CREBBP
SCHEMBL3044637 0.87 NR1H2 (0.39) NR1H2NR1H3TBK1
SCHEMBL3039181 0.86 NR1H2 (0.36) NR1H2BRD4CREBBPNR1H3TBK1
SCHEMBL3048520 0.86 NR1H2 (0.38) NR1H2ATRATRIPBRD4CREBBP
SCHEMBL3047413 0.86 NR1H2 (0.36) NR1H2ATRATRIPBRD4CREBBP
SCHEMBL3048979 0.86 NR1H2 (0.36) NR1H2ATRATRIPBRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed