SCHEMBL5048844

SCHEMBL5048844

CCOC(=O)CN(C(C)=Cc1cc(F)ccc1F)C1CCN(CCN2C(=O)COc3ccc(C#N)cc32)CC1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.41
USP2 O75604 1/20 0.39
HTT P42858 1/20 0.39
CHRM1 P11229 5/20 0.37
CHRM5 P08912 1/20 0.37
CHRM3 P20309 1/20 0.37
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
THRB P10828 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL708746 0.87 KCNH2 (0.41) KCNH2USP2HTTCHRM1CHRM5
SCHEMBL708745 0.87 KCNH2 (0.41) KCNH2USP2HTTCHRM1CHRM5
SCHEMBL706228 0.74 KCNH2 (0.55) KCNH2CHRM1CHRM5CHRM3
SCHEMBL706227 0.74 KCNH2 (0.55) KCNH2CHRM1CHRM5CHRM3
SCHEMBL921491 0.72 KCNH2 (0.61) KCNH2CHRM1CHRM5CHRM3CYP3A4
SCHEMBL705187 0.71 KCNH2 (0.53) KCNH2HTTCHRM1CHRM5CHRM3
SCHEMBL708349 0.69 KCNH2 (0.59) KCNH2CHRM1CYP3A4CYP2C9CYP2C19
SCHEMBL706005 0.69 KCNH2 (0.56) KCNH2CHRM1CHRM5CHRM3DRD2
Trifluoroacetic Acid SCHEMBL708560 0.68 KCNH2 (0.53) KCNH2CHRM1CHRM5CHRM3CYP3A4
SCHEMBL707478 0.68 CHRM1 (0.39) KCNH2CHRM1CHRM5CHRM3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893599-A1 COMPOUNDS FOR THE TREATMENT OF MULTI-DRUG RESISTANT BACTERIAL INFECTIONS AstraZeneca AB (SE) 2008-03-05 EP claimed
WO-2006134378-A1 COMPOUNDS FOR THE TREATMENT OF MULTI-DRUG RESISTANT BACTERIAL INFECTIONS ASTRAZENECA AB (SE) 2006-12-21 WO claimed